The management of metastatic GIST: current standard and investigational therapeutics

CM Kelly, L Gutierrez Sainz, P Chi - Journal of Hematology & Oncology, 2021‏ - Springer
Gastrointestinal stromal tumor (GIST) is the most common mesenchymal tumor of the
gastrointestinal tract. The majority of GISTs harbor gain of function mutations in either KIT or …

[HTML][HTML] Tropomyosin receptor kinase (TRK) biology and the role of NTRK gene fusions in cancer

A Amatu, A Sartore-Bianchi, K Bencardino… - Annals of …, 2019‏ - Elsevier
The tropomyosin receptor kinase (TRK) family of receptor tyrosine kinases are encoded by
NTRK genes and have a role in the development and normal functioning of the nervous …

Gastrointestinal stromal tumours: ESMO–EURACAN–GENTURIS Clinical Practice Guidelines for diagnosis, treatment and follow-up

PG Casali, JY Blay, N Abecassis, J Bajpai, S Bauer… - Annals of oncology, 2022‏ - Elsevier
Highlights•This clinical practice guideline provides key recommendations on the
management of gastrointestinal stromal tumours.•Recommendations have been agreed …

The ETS family of oncogenic transcription factors in solid tumours

GM Sizemore, JR Pitarresi, S Balakrishnan… - Nature Reviews …, 2017‏ - nature.com
Findings over the past decade have identified aberrant activation of the ETS transcription
factor family throughout all stages of tumorigenesis. Specifically in solid tumours, gene …

NCCN Guidelines® Insights: Gastrointestinal Stromal Tumors, Version 2.2022: Featured Updates to the NCCN Guidelines

M von Mehren, JM Kane, RF Riedel, JK Sicklick… - Journal of the National …, 2022‏ - jnccn.org
Gastrointestinal stromal tumors (GIST) are the most common type of soft tissue sarcoma that
occur throughout the gastrointestinal tract. Most of these tumors are caused by oncogenic …

Gastrointestinal stromal tumor: challenges and opportunities for a new decade

C Serrano, S George - Clinical Cancer Research, 2020‏ - AACR
Gastrointestinal stromal tumor (GIST) provides a paradigm to evaluate new molecularly
targeted therapies and to identify structural and functional mechanisms for drug response …

[HTML][HTML] JSCO—ESMO—ASCO—JSMO—TOS: international expert consensus recommendations for tumour-agnostic treatments in patients with solid tumours with …

T Yoshino, G Pentheroudakis, S Mishima… - Annals of …, 2020‏ - Elsevier
Highlights•The PD-1 antibody pembrolizumab and the TRK inhibitors larotrectinib and
entrectinib recently received regulatory approval.•Such tumour-agnostic regulatory …

[HTML][HTML] Prognostic indicators for gastrointestinal stromal tumors: a review

H Zhang, Q Liu - Translational Oncology, 2020‏ - Elsevier
Gastrointestinal stromal tumors (GISTs) are potentially malignancies that can occur
anywhere in the digestive tract. Tyrosine kinase inhibitors (TKIs) such as imatinib have …

A review of NTRK fusions in cancer

CA Manea, DC Badiu, IC Ploscaru… - Annals of Medicine …, 2022‏ - journals.lww.com
The family of the neurotrophic tropomyosin kinase receptors (NTRK or TRK) is a part of the
transmembrane tyrosine kinases responsible for neuronal development. The members of …

FGFR1 and NTRK3 actionable alterations in “Wild-Type” gastrointestinal stromal tumors

E Shi, J Chmielecki, CM Tang, K Wang… - Journal of translational …, 2016‏ - Springer
Abstract Background About 10–15% of adult, and most pediatric, gastrointestinal stromal
tumors (GIST) lack mutations in KIT, PDGFRA, SDHx, or RAS pathway components (KRAS …