Challenges of peptide and protein drug delivery by oral route: Current strategies to improve the bioavailability

S Verma, UK Goand, A Husain… - Drug development …, 2021 - Wiley Online Library
Advancement in biotechnology provided a notable expansion of peptide and protein
therapeutics, used as antigens, vaccines, hormones. It has a prodigious potential to treat a …

Microneedle mediated transdermal delivery of protein, peptide and antibody based therapeutics: current status and future considerations

M Kirkby, ARJ Hutton, RF Donnelly - Pharmaceutical Research, 2020 - Springer
The success of protein, peptide and antibody based therapies is evident-the
biopharmaceuticals market is predicted to reach $388 billion by 2024 [1], and more than half …

Dual functionalized liposome-mediated gene delivery across triple co-culture blood brain barrier model and specific in vivo neuronal transfection

B dos Santos Rodrigues, H Oue, A Banerjee… - Journal of controlled …, 2018 - Elsevier
Gene therapy has become a promising approach for neurodegenerative disease treatment,
however there is an urgent need to develop an efficient gene carrier to transport gene …

[HTML][HTML] Use of protamine in nanopharmaceuticals—a review

I Ruseska, K Fresacher, C Petschacher, A Zimmer - Nanomaterials, 2021 - mdpi.com
Macromolecular biomolecules are currently dethroning classical small molecule
therapeutics because of their improved targeting and delivery properties. Protamine-a small …

Surface modification of lipid-based nanocarriers for cancer cell-specific drug targeting

CH Kim, SG Lee, MJ Kang, S Lee, YW Choi - Journal of Pharmaceutical …, 2017 - Springer
Targeted drug delivery systems using nanocarriers for anticancer drugs have been
investigated for over several decades. Among the many nanocarrier systems, lipid-based …

Novel strategies in the oral delivery of antidiabetic peptide drugs–Insulin, GLP 1 and its analogs

R Ismail, I Csóka - European journal of pharmaceutics and …, 2017 - Elsevier
As diabetes is a complex disorder being a major cause of mortality and morbidity in
epidemic rates, continuous research has been done on new drug types and administration …

Bile acid transporter-mediated oral absorption of insulin via hydrophobic ion-pairing approach

S Bashyal, JE Seo, YW Choi, S Lee - Journal of Controlled Release, 2021 - Elsevier
Despite many ongoing and innovative approaches, there are still formidable challenges in
the clinical translation of oral peptide drugs into marketable products due to their low …

Effect of the lipid landscape on the efficacy of cell-penetrating peptides

F Zakany, IM Mándity, Z Varga, G Panyi, P Nagy… - Cells, 2023 - mdpi.com
Every cell biological textbook teaches us that the main role of the plasma membrane is to
separate cells from their neighborhood to allow for a controlled composition of the …

Development and screening of brain-targeted lipid-based nanoparticles with enhanced cell penetration and gene delivery properties

B dos Santos Rodrigues, S Lakkadwala… - International journal …, 2019 - Taylor & Francis
Background The potential of gene therapy for treatment of neurological disorders can be
explored using designed lipid-based nanoparticles such as liposomes, which have …

Critical material designs for mucus-and mucosa-penetrating oral insulin nanoparticle development

Y Zaiki, LY Lim, TW Wong - International Materials Reviews, 2023 - journals.sagepub.com
Subcutaneous and pulmonary insulin is associated with medical and pharmaceutical
complications. Oral insulin mimics physiological glucose regulation with reduced …