From antibacterial to antitumour agents: a brief review on the chemical and medicinal aspects of sulfonamides
H Azevedo-Barbosa, DF Dias, LL Franco… - Mini Reviews in …, 2020 - ingentaconnect.com
Sulfonamides have been in clinical use for many years, and the development of bioactive
substances containing the sulfonamide subunit has grown steadily in view of their important …
substances containing the sulfonamide subunit has grown steadily in view of their important …
Dithiol proteins as guardians of the intracellular redox milieu in parasites: old and new drug targets in trypanosomes and malaria‐causing plasmodia
RL Krauth‐Siegel, H Bauer… - Angewandte Chemie …, 2005 - Wiley Online Library
Parasitic diseases such as slee** sickness, Chagas' heart disease, and malaria are major
health problems in poverty‐stricken areas. Antiparasitic drugs that are not only active but …
health problems in poverty‐stricken areas. Antiparasitic drugs that are not only active but …
Quantum computational, spectroscopic investigations on N-(2-((2-chloro-4, 5-dicyanophenyl) amino) ethyl)-4-methylbenzenesulfonamide by DFT/TD-DFT with …
The experimental (x-ray, FT-IR NMR and UV-Vis. Spectral data) and theoretical researches
of N-(2-((2-chloro-4, 5-dicyanophenyl) amino) ethyl)-4-methylbenzenesulfonamide molecule …
of N-(2-((2-chloro-4, 5-dicyanophenyl) amino) ethyl)-4-methylbenzenesulfonamide molecule …
[LIVRE][B] Side reactions in Organic Synthesis: a guide to successful synthesis design
FZ Dörwald - 2006 - books.google.com
Most syntheses in the chemical research laboratory fail and usually require several attempts
before proceeding satisfactorily. Failed syntheses are not only discouraging and frustrating …
before proceeding satisfactorily. Failed syntheses are not only discouraging and frustrating …
“Recycling” classical drugs for malaria
Malaria has been a human health concern ever since the dawn of mankind, but despite the
huge struggles made to date to fight this infection, in 2012 over half a million people were …
huge struggles made to date to fight this infection, in 2012 over half a million people were …
Antibacterial metal complexes of o‐sulfamoylbenzoic acid: Synthesis, characterization, and DFT study
Herein, antibacterial transition metal complexes of ML2 type having o‐sulfamoylbenzoic
acid as ligand were synthesized from saccharin. All characterization techniques confirmed …
acid as ligand were synthesized from saccharin. All characterization techniques confirmed …
[PDF][PDF] Biological activity and synthesis of sulfonamide derivatives: a brief review
A Kołaczek, I Fusiarz, J Ławecka, D Branowska - Chemik, 2014 - researchgate.net
Sulfonamides (sulfa drugs) were the first drugs largely employed and systematically used as
preventive and chemotherapeutic agents against various diseases [1]. Over 30 drugs …
preventive and chemotherapeutic agents against various diseases [1]. Over 30 drugs …
Design, synthesis, ADME prediction and pharmacological evaluation of novel benzimidazole-1, 2, 3-triazole-sulfonamide hybrids as antimicrobial and antiproliferative …
Background Nitrogen heterocyclic rings and sulfonamides have attracted attention of several
researchers. Results A series of regioselective imidazole-based mono-and bis-1, 4 …
researchers. Results A series of regioselective imidazole-based mono-and bis-1, 4 …
Biological evaluation of some new N-(2, 6-dimethoxypyrimidinyl) thioureido benzenesulfonamide derivatives as potential antimicrobial and anticancer agents
A series of novel heterocyclic thioureas 3a-u containing sulfonamide moiety have been
synthesized by the condensation of isothiocyanatobenzenesulfonamide 2 with a variety of …
synthesized by the condensation of isothiocyanatobenzenesulfonamide 2 with a variety of …
Synthesis of Benzimidazole‐Sulfonyl Derivatives and Their Biological Activities
E Mulugeta, Y Samuel - Biochemistry Research International, 2022 - Wiley Online Library
Currently, the synthesis of new compounds with potential bioactivities has become a central
issue in the drug discovery arena. Among these new compounds, benzimidazole‐sulfonyl …
issue in the drug discovery arena. Among these new compounds, benzimidazole‐sulfonyl …