[HTML][HTML] Bioavailability enhancement techniques for poorly aqueous soluble drugs and therapeutics

DV Bhalani, B Nutan, A Kumar, AK Singh Chandel - Biomedicines, 2022‏ - mdpi.com
The low water solubility of pharmacoactive molecules limits their pharmacological potential,
but the solubility parameter cannot compromise, and so different approaches are employed …

Pharmaceutical dispersion techniques for dissolution and bioavailability enhancement of poorly water-soluble drugs

X Zhang, H **ng, Y Zhao, Z Ma - Pharmaceutics, 2018‏ - mdpi.com
Over the past decades, a large number of drugs as well as drug candidates with poor
dissolution characteristics have been witnessed, which invokes great interest in enabling …

[HTML][HTML] The potential use of simvastatin for cancer treatment: A review

JA Duarte, ALB de Barros, EA Leite - Biomedicine & Pharmacotherapy, 2021‏ - Elsevier
Statins, typically used to reduce lipid levels, have been rediscovered for exhibiting
anticancer activities. Among them, especially simvastatin may influence the proliferation …

Use of transethosomes for enhancing the transdermal delivery of olmesartan medoxomil: in vitro, ex vivo, and in vivo evaluation

R Albash, AA Abdelbary, H Refai… - International journal of …, 2019‏ - Taylor & Francis
Introduction and aim Olmesartan medoxomil (OLM) is an antihypertensive drug with low oral
bioavailability due to extensive first-pass metabolism. This study aimed to prepare transetho …

Methods for preparation of nanostructured lipid carriers

E Gomaa, HA Fathi, NG Eissa, M Elsabahy - Methods, 2022‏ - Elsevier
Construction of nanocarriers of different structures and properties have shown great promise
as delivery systems for a wide range of drugs to improve therapeutic effects and reduce side …

Recent progress in Zein nanoparticles: a promising approach for advancing Cancer therapy

MS Khan, M Fatima, G Gupta, S Md… - Journal of Drug Delivery …, 2024‏ - Elsevier
A holistic approach is now necessary in cancer research to address the patients' discomfort
and alleviate the shortcomings in chemotherapy treatment. Despite the existence of several …

Development of a nanostructured lipid carrier (NLC) by a low-energy method, comparison of release kinetics and molecular dynamics simulation

AC Ortiz, O Yañez, E Salas-Huenuleo, JO Morales - Pharmaceutics, 2021‏ - mdpi.com
Lipid nanocarriers have a great potential for improving the physicochemical characteristics
and behavior of poorly water-soluble drugs, such as aqueous dispersibility and oral …

[HTML][HTML] Lipid-based nanoparticles: Enhanced cellular uptake via surface thiolation

P Knoll, GF Racaniello, V Laquintana, F Veider… - International Journal of …, 2023‏ - Elsevier
The aim of this study was to evaluate the uptake mechanism of thiolated nanostructured lipid
carriers (NLCs). NLCs were decorated with a short-chain polyoxyethylene (10) stearyl ether …

[HTML][HTML] Nanomedicine-based disulfiram and metal ion co-delivery strategies for cancer treatment

X Shen, H Sheng, Y Zhang, X Dong, L Kou… - International Journal of …, 2024‏ - Elsevier
Disulfiram (DSF) is a second-line drug for the clinical treatment of alcoholism and has long
been proven to be safe for use in clinical practice. In recent years, researchers have …

Bile salt stabilized nanovesicles as a promising drug delivery technology: A general overview and future perspectives

R Abdel-moneum, RS Abdel-Rashid - Journal of drug delivery science and …, 2023‏ - Elsevier
Bile salts stabilized nanovesicles (bilosomes) have received tremendous attention in the
previous decade due to their vast preferabilities as well as the flexibility of their modification …