Quality-by-design-based development of rivaroxaban-loaded liquisolid compact tablets with improved biopharmaceutical attributes

P Shah, H Desai, B Vyas, M Lalan, M Kulkarni - AAPS PharmSciTech, 2023 - Springer
Rivaroxaban (RXN) finds use in the management of pulmonary embolism and deep vein
thrombosis. Its poor solubility (5–7 µg/mL) and P-gp-mediated efflux from intestinal lining …

Discerning computational, in vitro and in vivo investigations of self-assembling empagliflozin polymeric micelles in type-2 diabetes

P Wagh, S Savaliya, B Joshi, B Vyas… - Drug Delivery and …, 2024 - Springer
Background Empagliflozin (EMPA) is an SGLT2 inhibitor, a new class of anti-diabetic
medication, indicated for treating type-2 diabetes. Its low permeability, poor solubility and …

A Review on Different Solubility Enhancement Techniques of Ticagrelor.

A Srivastava, MA Khan, S Bedi… - International Journal of …, 2023 - search.ebscohost.com
Ticagrelor is a BCS class IV drug that inhibits platelet action by reversibly binding to the
P2Y12 receptor. One of the major challenges faced by the class IV (low solubility, low …

Amalgamation of solid dispersion and melt adsorption techniques for augmentation of oral bioavailability of novel anticoagulant rivaroxaban

PJ Shah, MP Patel, J Shah, AB Nair, S Kotta… - Drug Delivery and …, 2022 - Springer
The objective of the present study was to evaluate the potential of solid dispersion adsorbate
(SDA) to improve the solubility and bioavailability of rivaroxaban (RXN). SDA of RXN was …

[HTML][HTML] Bioanalytical method development, in-vivo pharmacokinetic evaluation, ex-vivo platelet aggregation inhibition activity of a novel solid dispersion formulation of …

A Srivastava, S Bedi, AK Mehata… - Frontiers in Medical …, 2025 - pmc.ncbi.nlm.nih.gov
Background Ticagrelor, a potential antithrombotic drug indicated for cardiovascular events
with acute coronary syndrome, has been restricted from its oral use due to poor aqueous …

Amalgam of ternary solid dispersion and P-gp efflux inhibition in development of colon-targeted tablets of rifaximin

MS Lalan, PJ Shah, R Kadam… - Journal of Reports in …, 2022 - journals.lww.com
Background: Rifaximin, a BCS class IV drug, possesses low bioavailability due to low
solubility and low permeability attributable to P-gp efflux. The studies attempted to develop …

[PDF][PDF] Design, optimization, and characterization of a novel amorphous solid dispersion formulation for enhancement of solubility and dissolution of ticagrelor

A SRIVASTAVA, MA KHAN, S BEDI, U Bhandari - Int J App Pharm, 2023 - academia.edu
DESIGN, OPTIMIZATION, AND CHARACTERIZATION OF A NOVEL AMORPHOUS SOLID
DISPERSION FORMULATION FOR ENHANCEMENT OF SOLUBILITY AND D Page 1 DESIGN …

Fabrication of ticagrelor bioadhesive solid dispersion based on coaxial electrostatic spray to improve drug release and enhance oral bioavailability.

H Liu, H Zhang, C Gu, X Chen, Y Feng… - Pakistan Journal of …, 2023 - search.ebscohost.com
Due to the low solubility and poor bioavailability of Ticagrelor (TIC), the current study
developed a structured bioadhesive core-shell drug delivery system to address it. Ticagreior …