Machine learning methods for small data challenges in molecular science

B Dou, Z Zhu, E Merkurjev, L Ke, L Chen… - Chemical …, 2023 - ACS Publications
Small data are often used in scientific and engineering research due to the presence of
various constraints, such as time, cost, ethics, privacy, security, and technical limitations in …

Deep learning methods for molecular representation and property prediction

Z Li, M Jiang, S Wang, S Zhang - Drug Discovery Today, 2022 - Elsevier
Highlights•The deep learning method could effectively represent the molecular structure and
predict molecular property through diversified models.•One, two, and three-dimensional …

DeepPROTACs is a deep learning-based targeted degradation predictor for PROTACs

F Li, Q Hu, X Zhang, R Sun, Z Liu, S Wu, S Tian… - Nature …, 2022 - nature.com
The rational design of PROTACs is difficult due to their obscure structure-activity
relationship. This study introduces a deep neural network model-DeepPROTACs to help …

Transition state theory-inspired neural network for estimating the viscosity of deep eutectic solvents

LY Yu, GP Ren, XJ Hou, KJ Wu, Y He - ACS central science, 2022 - ACS Publications
The lack of accurate methods for predicting the viscosity of solvent materials, especially
those with complex interactions, remains unresolved. Deep eutectic solvents (DESs), an …

[HTML][HTML] A machine learning framework to trace tumor tissue-of-origin of 13 types of cancer based on DNA somatic mutation

B He, C Dai, J Lang, P Bing, G Tian, B Wang… - Biochimica et Biophysica …, 2020 - Elsevier
Carcinoma of unknown primary (CUP), defined as metastatic cancers with unknown cancer
origin, occurs in 3‐5 per 100 cancer patients in the United States. Heterogeneity and …

A review of deep learning-based approaches for detection and diagnosis of diverse classes of drugs

A Kumar, N Kumar, J Kuriakose, Y Kumar - Archives of Computational …, 2023 - Springer
Artificial intelligence-based drug discovery has gained attention lately since it drastically cuts
the time and money needed to produce new treatments. In recent years, a vast quantity of …

A general use QSAR-ARX model to predict the corrosion inhibition efficiency of drugs in terms of quantum mechanical descriptors and experimental comparison for …

C Beltran-Perez, AAA Serrano, G Solís-Rosas… - International Journal of …, 2022 - mdpi.com
A study of 250 commercial drugs to act as corrosion inhibitors on steel has been developed
by applying the quantitative structure-activity relationship (QSAR) paradigm. Hard-soft acid …

Alkaloids in contemporary drug discovery to meet global disease needs

S Daley, GA Cordell - Molecules, 2021 - mdpi.com
An overview is presented of the well-established role of alkaloids in drug discovery, the
application of more sustainable chemicals, and biological approaches, and the …

Pushing the boundaries of molecular property prediction for drug discovery with multitask learning BERT enhanced by SMILES enumeration

XC Zhang, CK Wu, JC Yi, XX Zeng, CQ Yang, AP Lu… - Research, 2022 - spj.science.org
Accurate prediction of pharmacological properties of small molecules is becoming
increasingly important in drug discovery. Traditional feature-engineering approaches …

Convolutional neural networks (CNNs): Concepts and applications in pharmacogenomics

JM Vaz, S Balaji - Molecular diversity, 2021 - Springer
Convolutional neural networks (CNNs) have been used to extract information from various
datasets of different dimensions. This approach has led to accurate interpretations in several …