Imidazo [1, 2‐a] pyridine is a well‐known scaffold in many marketed drugs, such as
Zolpidem, Minodronic acid, Miroprofen and DS‐1 and it also serves as a broadly applied …

We report a ruthenium-catalyzed tandem Guerbet–alkylation strategy for the valorization of
ethanol. The products of ethanol upgrading (higher-order alcohols) undergo subsequent C …

Scaffold-generating transformations of the Groebke-Blackburn-Bienaymé (GBB) reaction
products are reviewed. The literature cases were grouped according to the reactions …

Herein we report the development of a sequential synthesis route towards annulated
imidazo [4, 5-c] isoquinolines comprising a GBB-3CR, followed by an intramolecular …

A concise and efficient one-pot synthesis of novel N-fused tricyclic derivatives has been
developed by using the Groebke–Blackburn–Bienaymé (GBB) reaction, which involved the …

Abstract The Groebke–Blackburn–Bienaymé (GBB) three-component reaction, discovered in
1998, is a very efficient strategy to assemble imidazo [1, 2-a]-heterocycles starting from …

β-Carboline containing alkaloids are ubiquitously present in Nature, while imidazo [1, 2-a]
pyridine nucleus is incorporated in various synthetic commercial drugs and biologically …

A facile and efficient protocol has been unfolded towards the diversity-oriented synthesis of
highly fluorescent pyrazole C-3 (5) tethered imidazo [1, 2-a] azines via an La (OTf) 3 …

Chloro-3-formyl quinoline has been applied as an aldehyde moiety in the Groebke–
Blackburn–Bienaymé multi-component reaction with isocyanides, 2-aminoazines, and 2 …

In this work, we continue our adventure in the chemistry of 5-5 tri-nitrogen bicycles. We
disclose herein a one-step reaction to synthesize 1H-imidazo [1, 5-a] imidazoles with …