PI3K/Akt/mTOR inhibitors in cancer: At the bench and bedside

AS Alzahrani - Seminars in cancer biology, 2019 - Elsevier
Abstract Phosphatidylinositol 3-kinase (PI3K)/Akt/mammalian target of rapamycin (mTOR)
signaling pathway is one of the major cellular signaling pathways that plays an important …

Targeting Akt in cancer for precision therapy

H Hua, H Zhang, J Chen, J Wang, J Liu… - Journal of Hematology & …, 2021 - Springer
Biomarkers-guided precision therapeutics has revolutionized the clinical development and
administration of molecular-targeted anticancer agents. Tailored precision cancer therapy …

[HTML][HTML] PI3K/AKT/mTOR-targeted therapy for breast cancer

K Zhu, Y Wu, P He, Y Fan, X Zhong, H Zheng, T Luo - Cells, 2022 - mdpi.com
Phosphatidylinositol 3-kinase (PI3K), protein kinase B (PKB/AKT) and mechanistic target of
rapamycin (mTOR)(PAM) pathways play important roles in breast tumorigenesis and confer …

AKT inhibitors: new weapons in the fight against breast cancer?

F Martorana, G Motta, G Pavone, L Motta… - Frontiers in …, 2021 - frontiersin.org
The serine/threonine kinase AKT is a key component of the PI3K/AKT/mTOR signaling
pathway as it exerts a pivotal role in cell growth, proliferation, survival, and metabolism …

Targeting AKT for cancer therapy

M Shariati, F Meric-Bernstam - Expert opinion on investigational …, 2019 - Taylor & Francis
Introduction: Targeted therapies in cancer aim to inhibit specific molecular targets
responsible for enhanced tumor growth. AKT/PKB (protein kinase B) is a serine threonine …

ESR1 mutations in breast cancer

D Dustin, G Gu, SAW Fuqua - Cancer, 2019 - Wiley Online Library
The acquisition of ligand‐independent ESR1 mutations during aromatase inhibitor therapy
in metastatic estrogen receptor (ER)‐positive breast cancer is a common mechanism of …

Recent advances with precision medicine treatment for breast cancer including triple-negative sub-type

MA Subhan, F Parveen, H Shah, SSK Yalamarty… - Cancers, 2023 - mdpi.com
Simple Summary The progress of next-generation sequencing technologies has raised
huge expectations for precision-medicine therapy approaches in breast cancer and triple …

Phase II trial of AKT inhibitor MK-2206 in patients with advanced breast cancer who have tumors with PIK3CA or AKT mutations, and/or PTEN loss/PTEN mutation

Y **ng, NU Lin, MA Maurer, H Chen, A Mahvash… - Breast Cancer …, 2019 - Springer
Abstract Background The PI3K/AKT pathway is activated through PIK3CA or AKT1 mutations
and PTEN loss in breast cancer. We conducted a phase II trial with an allosteric AKT …

[HTML][HTML] Targeting autophagy-related protein kinases for potential therapeutic purpose

H **ang, J Zhang, C Lin, L Zhang, B Liu… - … Pharmaceutica Sinica B, 2020 - Elsevier
Autophagy, defined as a scavenging process of protein aggregates and damaged
organelles mediated by lysosomes, plays a significant role in the quality control of …

Akt-targeted therapy as a promising strategy to overcome drug resistance in breast cancer–A comprehensive review from chemotherapy to immunotherapy

PJ Kaboli, F Salimian, S Aghapour, S **ang… - Pharmacological …, 2020 - Elsevier
Breast cancer is the most frequently occurring cancer in women. Chemotherapy in
combination with immunotherapy has been used to treat breast cancer. Atezolizumab …