[PDF][PDF] Benzimidazole derivatives–an overview

R Walia, M Hedaitullah, SF Naaz… - Int. J. Res. Pharm …, 2011 - cmapspublic3.ihmc.us
Benzimidazole derivatives play important role in medical field with so many
Pharmacological activities such as antimicrobial, antiviral, antidiabetic and anticancer …

Antimicrobial activity and a SAR study of some novel benzimidazole derivatives bearing hydrazone moiety

Y Özkay, Y Tunalı, H Karaca, İ Işıkdağ - European journal of medicinal …, 2010 - Elsevier
In this study 12 novel benzimidazole compounds bearing hydrazone moiety were
synthesized in order to investigate their possible antibacterial and antifungal activity …

Pyrazole carbohydrazide derivatives of pharmaceutical interest

LRS Dias, RRS Salvador - Pharmaceuticals, 2012 - mdpi.com
Pharmaceuticals | Free Full-Text | Pyrazole Carbohydrazide Derivatives of Pharmaceutical
Interest Next Article in Journal Comparison of Intraocular Pressure, Blood Pressure, Ocular …

Antibacterial and antifungal activities of new pyrazolo [3, 4-d] pyridazin derivatives

E Akbas, I Berber - European Journal of Medicinal Chemistry, 2005 - Elsevier
Several new pyrazolo [3, 4-d] pyridazin derivatives were prepared by the reaction of two new
1H-pyrazole-3-carboxylic acids and various hydrazines. The compounds were tested for …

Synthesis, structure optimization and antifungal screening of novel tetrazole ring bearing acyl-hydrazones

MA Malik, SA Al-Thabaiti, MA Malik - International journal of molecular …, 2012 - mdpi.com
Azoles are generally fungistatic, and resistance to fluconazole is emerging in several fungal
pathogens. In an attempt to find novel azole antifungal agents with improved activity, a …

Synthesis, in silico experiments and biological evaluation of 1, 3, 4-trisubstituted pyrazole derivatives as antimalarial agents

AA Bekhit, MN Saudi, AMM Hassan, SM Fahmy… - European journal of …, 2019 - Elsevier
Abstract New 1, 3, 4-trisubstituted pyrazole derivatives were synthesized and evaluated for
their antiplasmodial activity. Compounds 4b, 4c, 7a and 7d were the most potent …

Synthesis and antibacterial activity of 4-benzoyl-1-methyl-5-phenyl-1H-pyrazole-3-carboxylic acid and derivatives

E Akbas, I Berber, A Sener, B Hasanov - Il Farmaco, 2005 - Elsevier
Some new 1H-pyrazole-3-carboxylic acid and pyridazinone derivatives were synthesized
and evaluated for their antibacterial activities against Bacillus cereus ATCC 7064 …

[PDF][PDF] Synthesis of some new azoles with antiviral potential

AR Farghaly, H El-Kashef - Arkivoc, 2006 - academia.edu
Synthesis of some new azoles with antiviral potential Page 1 General Papers ARKIVOC
2006 (xi) 76-90 ISSN 1424-6376 Page 76 © ARKAT Synthesis of some new azoles with …

Antimicrobial activity of a new series of benzimidazole derivatives

Y Özkay, Y Tunalı, H Karaca, İ Işıkdağ - Archives of pharmacal research, 2011 - Springer
Due to antimicrobial importance of benzimidazoles and hydrazones, some
benzimidazolehydrazone compounds were synthesized to screen their antimicrobial activity …

The first-in-class pyrazole-based dual InhA-VEGFR inhibitors towards integrated antitubercular host-directed therapy

MM Shaaban, M Teleb, HM Ragab, M Singh… - Bioorganic …, 2024 - Elsevier
Several facets of the host response to tuberculosis have been tapped for clinical
investigation, especially targeting angiogenesis mediated by VEGF signaling from infected …