Lactate dehydrogenase A: A key player in carcinogenesis and potential target in cancer therapy

Y Feng, Y **ong, T Qiao, X Li, L Jia, Y Han - Cancer medicine, 2018‏ - Wiley Online Library
Elevated glycolysis remains a universal and primary character of cancer metabolism, which
deeply depends on dysregulated metabolic enzymes. Lactate dehydrogenase A (LDHA) …

MYC, metabolism, and cancer

ZE Stine, ZE Walton, BJ Altman, AL Hsieh… - Cancer …, 2015‏ - aacrjournals.org
The MYC oncogene encodes a transcription factor, MYC, whose broad effects make its
precise oncogenic role enigmatically elusive. The evidence to date suggests that MYC …

Equivariant 3D-conditional diffusion model for molecular linker design

I Igashov, H Stärk, C Vignac, A Schneuing… - Nature Machine …, 2024‏ - nature.com
Fragment-based drug discovery has been an effective paradigm in early-stage drug
development. An open challenge in this area is designing linkers between disconnected …

Role of mitochondrial membrane potential and lactate dehydrogenase a in apoptosis

S Zaib, A Hayyat, N Ali, A Gul… - Anti-Cancer Agents in …, 2022‏ - benthamdirect.com
Apoptosis is a programmed cell death that occurs due to the production of several catabolic
enzymes. During this process, several morphological and biochemical changes occur in …

Targeting lactate dehydrogenase-a inhibits tumorigenesis and tumor progression in mouse models of lung cancer and impacts tumor-initiating cells

H **e, J Hanai, JG Ren, L Kats, K Burgess, P Bhargava… - Cell metabolism, 2014‏ - cell.com
The lactate dehydrogenase-A (LDH-A) enzyme catalyzes the interconversion of pyruvate
and lactate, is upregulated in human cancers, and is associated with aggressive tumor …

The biochemical and clinical perspectives of lactate dehydrogenase: an enzyme of active metabolism

AA Khan, KS Allemailem… - … Metabolic & Immune …, 2020‏ - ingentaconnect.com
Background: Lactate dehydrogenase (LDH) is a group of oxidoreductase isoenzymes
catalyzing the reversible reaction between pyruvate and lactate. The five isoforms of this …

Lactate dehydrogenase 5: an old friend and a new hope in the war on cancer

K Augoff, A Hryniewicz-Jankowska, R Tabola - Cancer letters, 2015‏ - Elsevier
A hallmark of most cancer cells is an altered metabolism involving a shift to aerobic
glycolysis with lactate production coupled with a higher uptake of glucose as the main …

Fragment-based drug discovery using NMR spectroscopy

MJ Harner, AO Frank, SW Fesik - Journal of biomolecular NMR, 2013‏ - Springer
Nuclear magnetic resonance (NMR) spectroscopy has evolved into a powerful tool for
fragment-based drug discovery over the last two decades. While NMR has been traditionally …

Fragment linking strategies for structure-based drug design

A Bancet, C Raingeval, T Lomberget… - Journal of medicinal …, 2020‏ - ACS Publications
Fragment-based drug discovery is a strategy widely used in both academia and
pharmaceutical companies to generate small-molecule protein inhibitors and drug …

Quinoline 3-sulfonamides inhibit lactate dehydrogenase A and reverse aerobic glycolysis in cancer cells

J Billiard, JB Dennison, J Briand, RS Annan, D Chai… - Cancer & …, 2013‏ - Springer
Background Most normal cells in the presence of oxygen utilize glucose for mitochondrial
oxidative phosphorylation. In contrast, many cancer cells rapidly convert glucose to lactate in …