Targeting multidrug resistance-associated protein 1 (MRP1)-expressing cancers: Beyond pharmacological inhibition

KM Hanssen, M Haber, JI Fletcher - Drug Resistance Updates, 2021 - Elsevier
Resistance to chemotherapy remains one of the most significant obstacles to successful
cancer treatment. While inhibiting drug efflux mediated by ATP-binding cassette (ABC) …

ABCG2: determining its relevance in clinical drug resistance

RW Robey, O Polgar, J Deeken, KW To… - Cancer and Metastasis …, 2007 - Springer
Multidrug resistance is a major obstacle to successful cancer treatment. One mechanism by
which cells can become resistant to chemotherapy is the expression of ABC transporters that …

Mechanisms of multidrug resistance in cancer

JP Gillet, MM Gottesman - Multi-drug resistance in cancer, 2010 - Springer
The development of multidrug resistance (MDR) to chemotherapy remains a major
challenge in the treatment of cancer. Resistance exists against every effective anticancer …

Role of ABCG2/BCRP in biology and medicine

P Krishnamurthy, JD Schuetz - Annu. Rev. Pharmacol. Toxicol., 2006 - annualreviews.org
▪ Abstract The protein variously named ABCG2/BCRP/MXR/ABCP is a recently described
ATP-binding cassette (ABC) transporter originally identified by its ability to confer drug …

MRP1 and its role in anticancer drug resistance

JF Lu, D Pokharel, M Bebawy - Drug metabolism reviews, 2015 - Taylor & Francis
The phenomenon of multidrug resistance (MDR) in cancer is associated with the
overexpression of the ATP-binding cassette (ABC) transporter proteins, including multidrug …

Revisiting the ABCs of multidrug resistance in cancer chemotherapy

AK Tiwari, K Sodani, CL Dai… - Current …, 2011 - ingentaconnect.com
The adenosine triphosphate binding cassette (ABC) transporters are one of the largest
transmembrane gene families in humans. The ABC transporters are present in a number of …

ABCG2: structure, function and role in drug response

O Polgar, RW Robey, SE Bates - Expert opinion on drug …, 2008 - Taylor & Francis
ABCG2 was discovered in multi-drug-resistant cancer cells, with the identification of
chemotherapeutic agents, such as mitoxantrone, flavopiridol, methotrexate and irinotecan as …

Photoactivated H2 Nanogenerator for Enhanced Chemotherapy of Bladder Cancer

R Sun, X Liu, G Li, H Wang, Y Luo, G Huang, X Wang… - ACS …, 2020 - ACS Publications
Hydrogen gas can mitigate oxidative stress in many diseases and is regarded to be safe and
free of side effects. Inspired by a metalloenzyme in a variety of microorganisms, here, we …

ABCG2: the key to chemoresistance in cancer stem cells?

Y An, WM Ongkeko - Expert opinion on drug metabolism & …, 2009 - Taylor & Francis
Multi-drug chemoresistance remains one of the most common reasons for chemotherapy
failure. The membrane transporter protein ABCG2/BCRP1 has been shown in vitro to …

Prognostic markers for bladder cancer: International Consensus Panel on bladder tumor markers

T Habuchi, M Marberger, MJ Droller, GP Hemstreet III… - Urology, 2005 - Elsevier
The International Consensus Panel on cytology and bladder tumor markers evaluated
markers that have the ability to predict tumor recurrence, progression, development of …