Gold (III) complexes in medicinal chemistry

PI da Silva Maia, VM Deflon, U Abram - Future medicinal chemistry, 2014 - Taylor & Francis
A number of gold (III) compounds has been designed with the objective of overcoming the
disadvantages associated with the platinum-based drugs for cancer treatment. Compounds …

Synthesis, characterization, and biological activity of some 2, 4-diketo esters containing dehydrozingerone fragment: DNA and protein binding study

K Mihajlović, N Joksimović, N Janković… - Bioorganic & Medicinal …, 2023 - Elsevier
Due to the increased resistance to antibiotics, in recent years there has been a growing
interest in the discovery of new antimicrobial agents from different sources. Bacteria that are …

[HTML][HTML] Square planar Au (III), Pt (II) and Cu (II) complexes with quinoline-substituted 2, 2′: 6′, 2 ″-terpyridine ligands: From in vitro to in vivo biological properties

K Choroba, B Machura, A Szlapa-Kula… - European Journal of …, 2021 - Elsevier
Cancer is the second leading cause of death worldwide. Cisplatin has challenged cancer
treatment; however, resistance and side effects hamper its use. New agents displaying …

Spectroscopy, electrochemistry and antiproliferative properties of Au (iii), Pt (ii) and Cu (ii) complexes bearing modified 2, 2′: 6′, 2′′-terpyridine ligands

A Maroń, K Czerwińska, B Machura, L Raposo… - Dalton …, 2018 - pubs.rsc.org
Structural, spectroscopic and electrochemical properties of six complexes [AuCl (L1)](PF6)
2· CH3CN (1),[AuCl (L2)](PF6) 2 (2),[PtCl (L1)](BPh4)· CH3CN (3),[PtCl (L2)](SO3CF3)(4) …

New gold pincer-type complexes: synthesis, characterization, DNA binding studies and cytotoxicity

S Radisavljević, I Bratsos, A Scheurer… - Dalton …, 2018 - pubs.rsc.org
With the aim of assessing whether Au (III) compounds with pincer type ligands might be
utilized as potential antitumor agents, three new monofunctional Au (III) complexes of the …

The synthesis, spectroscopic characterization and anticancer activity of new mono and binuclear phosphanegold (I) dithiocarbamate complexes

M Altaf, M Monim-ul-Mehboob, AA Isab… - New Journal of …, 2015 - pubs.rsc.org
A new series of mononuclear [t-Bu3PAuS2CN (C7H7) 2](1), and binuclear [(DPPM) Au2
(S2CN (CH3) 2) 2](2),[(DPPM) Au2 (S2CN (C2H5) 2) 2](3) and [(DPPM) Au2 (S2CN (C7H7) …

Anticancer activity and apoptosis induction of gold (III) complexes containing 2, 2′-bipyridine-3, 3′-dicarboxylic acid and dithiocarbamates

A Alhoshani, AAA Sulaiman, HMA Sobeai, W Qamar… - Molecules, 2021 - mdpi.com
Three novel gold (III) complexes (1–3) of general composition [Au (Bipydc)(S2CNR2)] Cl2
(Bipydc= 2, 2′-bipyridine-3, 3′-dicarboxylic acid and R= methyl for …

Cytotoxic gold (iii) complexes incorporating a 2, 2′: 6′, 2′′-terpyridine ligand framework–the impact of the substituent in the 4′-position of a terpy ring

K Czerwińska, M Golec, M Skonieczna… - Dalton …, 2017 - pubs.rsc.org
Two gold (III) complexes incorporating 2, 2′: 6′, 2′′-terpyridine derivatives have been
synthesised and characterized, and the possibility of tuning the cytotoxic activity by structural …

Impedance technology reveals correlations between cytotoxicity and lipophilicity of mono and bimetallic phosphine complexes

P Fonteh, A Elkhadir, B Omondi, I Guzei, J Darkwa… - Biometals, 2015 - Springer
Label free impedance technology enables the monitoring of cell response patterns post
treatment with drugs or other chemicals. Using this technology, a correlation between the …

Synthesis, characterization and in vitro cytotoxicity of gold (III) dialkyl/diaryldithiocarbamato complexes

M Altaf, AA Isab, J Vančo, Z Dvořák, Z Trávníček… - RSC …, 2015 - pubs.rsc.org
A series of six dialkyl/diaryldithiocarbamato (dtc) gold (III) complexes 1–6 of the composition
[Au (Me2dtc) 2] Cl (1),[Au (Me2dtc) Cl2](2),[Au (Et2dtc) 2] Cl (3),[Au (Et2dtc) Cl2](4),[Au …