Recent advances in the chemistry and biology of benzothiazoles

RK Gill, RK Rawal, J Bariwal - Archiv der Pharmazie, 2015 - Wiley Online Library
Benzothiazole is a privileged heterocyclic scaffold having a benzene ring fused with a five‐
membered thiazole ring. This moiety has attracted considerable attention because of its …

Biological aspects of emerging benzothiazoles: a short review

R Ali, N Siddiqui - Journal of chemistry, 2013 - Wiley Online Library
In recent years heterocyclic compounds analogues and derivatives have attracted wide
attention due to their useful biological and pharmacological properties. Benzothiazole is …

Curcumin-I Knoevenagel's condensates and their Schiff's bases as anticancer agents: synthesis, pharmacological and simulation studies

I Ali, A Haque, K Saleem, MF Hsieh - Bioorganic & medicinal chemistry, 2013 - Elsevier
Pyrazolealdehydes (4a–d), Knoevenagel's condensates (5a–d) and Schiff's bases (6a–d) of
curcumin-I were synthesized, purified and characterized. Hemolysis assays, cell line …

Curcumin based pyrazole-thiazole hybrids as antiproliferative agents: Synthesis, pharmacokinetic, photophysical properties, and docking studies

R Palabindela, R Guda, G Ramesh, R Bodapati… - Journal of Molecular …, 2023 - Elsevier
A series of new curcumin pyrazole-thiazole hybrids (C 1-C 8) were synthesized and
characterized by fundamental spectral analysis. The synthesized compounds were tested for …

The potency of heterocyclic curcumin analogues: An evidence-based review

FC Rodrigues, NVA Kumar, G Thakur - Pharmacological Research, 2021 - Elsevier
Curcumin, a potent phytochemical, has been a significant lead compound and has been
extensively investigated for its multiple bioactivities. Owing to its natural origin, non-toxic …

Design, synthesis, antifungal activity, and molecular docking studies of novel chiral isoxazoline-benzofuran-sulfonamide derivatives

Y Yan, A Bao, Y Wang, X **e, D Wang… - Journal of Agricultural …, 2024 - ACS Publications
Succinate dehydrogenase (SDH) is one of the most important molecular targets for the
development of novel fungicides. With the emerging problem of resistance in plant fungal …

Exploiting the biological efficacy of benzimidazole based Schiff base complexes with l-Histidine as a co-ligand: Combined molecular docking, DNA interaction …

G Kumaravel, PP Utthra, N Raman - Bioorganic chemistry, 2018 - Elsevier
Four new metal complexes were synthesized and screened for their cytotoxic activity after
sufficient assertion from the preliminary DNA binding studies. The metal complexes could …

Antioxidant activity and electrochemical elucidation of the enigmatic redox behavior of curcumin and its structurally modified analogues

NS Jha, S Mishra, SK Jha, A Surolia - Electrochimica Acta, 2015 - Elsevier
Here, we report studies on the antioxidant activity and redox behavior of curcumin and its
structurally modified synthetic analogues. We have synthesized a number of analogues of …

Importance of fluorine in benzazole compounds

T Al-Harthy, W Zoghaib, R Abdel-Jalil - Molecules, 2020 - mdpi.com
Fluorine-containing heterocycles continue to receive considerable attention due to their
unique properties. In medicinal chemistry, the incorporation of fluorine in small molecules …

Structure activity relationship, cytotoxicity and evaluation of antioxidant activity of curcumin derivatives

PK Sahu, PK Sahu, PL Sahu, DD Agarwal - Bioorganic & medicinal …, 2016 - Elsevier
Abstract Series of curcumin derivatives/analogues were designed and efficient method for
synthesis thereof is described. All the synthesized compounds have been screened for their …