The synthetic and therapeutic expedition of isoxazole and its analogs

N Agrawal, P Mishra - Medicinal Chemistry Research, 2018‏ - Springer
Isoxazole, constituting an important family of five-membered heterocycles with one oxygen
atom and one nitrogen atom at adjacent positions is of immense importance because of its …

Protein tyrosine phosphatase 1B (PTP1B) and obesity

H Cho - Vitamins & hormones, 2013‏ - Elsevier
Protein tyrosine phosphatase 1B (PTP1B) is a negative regulator of the leptin and insulin
signaling pathways. The important roles of PTP1B related to obesity and diabetes were …

Synthesis of isoxazoles by hypervalent iodine-induced cycloaddition of nitrile oxides to alkynes

AM Jawalekar, E Reubsaet, FPJT Rutjes… - Chemical …, 2011‏ - pubs.rsc.org
Treatment of oximes with hypervalent iodine leads to substituted isoxazolesvia rapid
formation of nitrile oxides. Reaction with terminal alkynes led to a series of 3, 5-disubstituted …

Aldose reductase and protein tyrosine phosphatase 1B inhibitors as a promising therapeutic approach for diabetes mellitus

A Kousaxidis, A Petrou, V Lavrentaki… - European Journal of …, 2020‏ - Elsevier
Diabetes mellitus is a metabolic disease characterized by high blood glucose levels and
usually associated with several chronic pathologies. Aldose reductase and protein tyrosine …

Synthesis of chalcones and flavanones using Julia–Kocienski olefination

A Kumar, S Sharma, VD Tripathi, S Srivastava - Tetrahedron, 2010‏ - Elsevier
A new application of Julia–Kocienski olefination for the synthesis of chalcones and
flavanones has been described. 2-(Benzo [d] thiazol-2-ylsulfonyl)-1-phenylethanones have …

Epihalohydrins in organic synthesis

GS Singh, K Mollet, M D'hooghe… - Chemical Reviews, 2013‏ - ACS Publications
Epihalohydrins [2-(halomethyl) oxiranes, 1, 2-epoxy-3-halopropanes](Figure 1) are well-
known versatile synthons and important reagents in the realm of organic synthesis …

Natural product inspired diversity oriented synthesis of tetrahydroquinoline scaffolds as antitubercular agent

A Kumar, S Srivastava, G Gupta… - ACS Combinatorial …, 2011‏ - ACS Publications
An efficient natural product inspired diversity oriented syn thesis of tetrahydroquinoline
analogues has been developed using the natural carbohydrate derived solid acid catalyst …

[HTML][HTML] Synthesis and biological evaluation of amide derivatives of isoxazole-imidazo [2, 1-b] thiazole as anticancer agents

KB Alapati, D Sravani, BBV Sailaja, B Saritha… - Results in Chemistry, 2024‏ - Elsevier
A new series of amide functionality contained isoxazole-imidazo [2, 1-b] thiazole (12a-j)
were synthesized and their structures were characterized by analytical techniques. Further …

Design and synthesis of 2, 4-disubstituted polyhydroquinolines as prospective antihyperglycemic and lipid modulating agents

A Kumar, S Sharma, VD Tripathi, RA Maurya… - Bioorganic & medicinal …, 2010‏ - Elsevier
A series of 2, 4-disubstituted polyhydroquinoline were synthesized and evaluated for their in
vivo antihyperglycemic as well as antidyslipidemic activities. Several synthesized …

Synthesis of multiply arylated heteroarenes, including bioactive derivatives, via palladium-catalyzed direct C–H arylation of heteroarenes with (pseudo) aryl halides or …

R Rossi, F Bellina, M Lessi, C Manzini, LA Perego - Synthesis, 2014‏ - thieme-connect.com
This review with 387 references covers the literature until the end of November 2013 on the
synthesis of multiply arylated heteroarenes via highly selective palladium-catalyzed direct C …