The rcdk and cluster R packages applied to drug candidate selection

A Voicu, N Duteanu, M Voicu, D Vlad… - Journal of …, 2020 - Springer
The aim of this article is to show how thevpower of statistics and cheminformatics can be
combined, in R, using two packages: rcdk and cluster. We describe the role of clustering …

3-Pyridinylidene derivatives of chemically modified lupane and ursane triterpenes as promising anticancer agents by targeting apoptosis

O Kazakova, C Șoica, M Babaev, A Petrova… - International Journal of …, 2021 - mdpi.com
Cancer persists as a global challenge due to the extent to which conventional anticancer
therapies pose high risks counterbalanced with their therapeutic benefit. Naturally occurring …

Design, Synthesis and Biological Activity Evaluation of S-Substituted 1H-5-Mercapto-1,2,4-Triazole Derivatives as Antiproliferative Agents in Colorectal Cancer

M Mioc, S Avram, V Bercean, L Kurunczi… - Frontiers in …, 2018 - frontiersin.org
Colon cancer is a widespread pathology with complex biochemical etiology based on a
significant number of intracellular signaling pathways that play important roles in …

Expression of E-cadherin in lung carcinoma, other than those with small cells (NSCLC).

ML Grigoraş, TS Arghirescu, R Folescu… - Romanian Journal of …, 2017 - europepmc.org
It was suggested that the decrease and/or loss of E-cadherin expression in non-small cell
lung cancer (NSCLC) is responsible for the development of the malignant phenotype …

Construction of a novel bispecific fusion protein to enhance targeting for pancreatic cancer imaging

Q Wang, H Yan, Z Wang, Z Li, D Li, Z Li, K Wang, J Tian… - Biomaterials, 2020 - Elsevier
Early detection and diagnosis are the most important endeavors for reducing associated
morbidity and mortality of pancreatic ductal adenocarcinoma (PDAC). Develo** molecular …

[PDF][PDF] S, oica

O Kazakova - Int. J. Mol. Sci, 2021 - academia.edu
Cancer persists as a global challenge due to the extent to which conventional anticancer
therapies pose high risks counterbalanced with their therapeutic benefit. Naturally occurring …

Synthesis, Cytotoxic Activity and Molecular Docking Studies of New Condensed Thieno[2,3-d]Pyrimidines as Antitumor Agents

S Kaliraj, R Jeyalakshmi, MK Kathiravan - Pharmaceutical Chemistry …, 2020 - Springer
A series of twenty molecules based on thienopyrimidine nucleus fused with 5-, 6-, and 7-
membered lactam rings as well as triazole were synthesized via 4-step reactions. The target …