Binding sites of anticancer drugs on human serum albumin (HSA): a review

P Molaei, H Mahaki, H Manoochehri… - Protein and peptide …, 2022 - benthamdirect.com
Background: To recognize the action of pharmacologically approved anticancer drugs in
biological systems, information regarding its pharmacokinetics, such as its transport within …

Vitamin k3 inhibits protein aggregation: implication in the treatment of amyloid diseases

P Alam, SK Chaturvedi, MK Siddiqi, RK Rajpoot… - Scientific reports, 2016 - nature.com
Protein misfolding and aggregation have been associated with several human diseases
such as Alzheimer's, Parkinson's and familial amyloid polyneuropathy etc. In this study, anti …

Spectrofluorimetric and molecular docking studies on the interaction of cyanidin-3-O-glucoside with whey protein, β-lactoglobulin

J Cheng, JH Liu, G Prasanna, P **g - International Journal of Biological …, 2017 - Elsevier
The interaction of β-Lactoglobulin (β-Lg) with cyanidin-3-O-glucoside (C3G) was
characterized using fluorescence, circular dichroism spectroscopy, and docking studies …

In vitro and in vivo inhibitory effect of anthocyanin-rich bilberry extract on α-glucosidase and α-amylase

Y Ji, D Liu, J Zhao, J Zhao, H Li, L Li, H Zhang, H Wang - Lwt, 2021 - Elsevier
The inhibition of glycosidase activity is regarded as an effective treatment for diabetes
mellitus. Bilberry (Vaccinium myrtillus L.) fruit has a high content of anthocyanins with …

Investigation of inhibitory potential of quercetin to the pyruvate dehydrogenase kinase 3: Towards implications in anticancer therapy

R Dahiya, T Mohammad, S Roy, S Anwar… - International journal of …, 2019 - Elsevier
Abstract Pyruvate dehydrogenase kinase 3 (PDK3) is a mitochondrial protein, has recently
been considered as a potential pharmacological target for varying types of cancer. Here, we …

Ascorbic acid inhibits human insulin aggregation and protects against amyloid induced cytotoxicity

P Alam, AZ Beg, MK Siddiqi, SK Chaturvedi… - Archives of biochemistry …, 2017 - Elsevier
Protein aggregation into oligomers and fibrils are associated with many human
pathophysiologies. Compounds that modulate protein aggregation and interact with …

Investigating the site selective binding of busulfan to human serum albumin: Biophysical and molecular docking approaches

M Siddiqi, S Nusrat, P Alam, S Malik… - International journal of …, 2018 - Elsevier
We have studied the binding of busulfan (BN) to human serum albumin (HSA) at
physiological pH 7.4 by using fluorescence, UV–vis and circular dichroism (CD) …

Investigation of the interaction between Chrysoeriol and xanthine oxidase using computational and in vitro approaches

Y Liu, C Han, T Lu, Y Liu, H Chen, C Yang, Y Tu… - International Journal of …, 2021 - Elsevier
Xanthine oxidase (XO) plays a vital role in inducing hyperuricemia and increasing the level
of superoxide free radicals in blood, and is proved as an important target for gout …

Discovery of 8-hydroxy-2-quinoline carbaldehyde derivatives as inhibitors for M1 aminopeptidase of leishmania donovani

J Kumar, R Qureshi, P Jagruthi, M Arifuddin… - International Journal of …, 2024 - Elsevier
M1 aminopeptidase is a metallopeptidase that plays a vital role in protein catabolism and
has been identified as a validated drug target in various parasites; however, our …

Anti-amyloidogenic behavior and interaction of diallylsulfide with human serum albumin

MK Siddiqi, P Alam, SK Chaturvedi, RH Khan - International journal of …, 2016 - Elsevier
In this work, binding of garlic component-Diallysulfide (DAS) with major human blood
transport protein, Human Serum Albumin (HSA) and its anti-amyloidogenic behavior has …