[HTML][HTML] From machine learning to deep learning: Advances of the recent data-driven paradigm shift in medicine and healthcare

C Chakraborty, M Bhattacharya, S Pal… - Current Research in …, 2024 - Elsevier
The medicine and healthcare sector has been evolving and advancing very fast. The
advancement has been initiated and shaped by the applications of data-driven, robust, and …

[HTML][HTML] Simulation-based approaches for drug delivery systems: Navigating advancements, opportunities, and challenges

I Salahshoori, M Golriz, MAL Nobre, S Mahdavi… - Journal of Molecular …, 2024 - Elsevier
Efficient drug delivery systems (DDSs) play a pivotal role in ensuring pharmaceuticals'
targeted and effective administration. However, the intricate interplay between drug …

Recent advances in machine-learning-based chemoinformatics: a comprehensive review

SK Niazi, Z Mariam - International Journal of Molecular Sciences, 2023 - mdpi.com
In modern drug discovery, the combination of chemoinformatics and quantitative structure–
activity relationship (QSAR) modeling has emerged as a formidable alliance, enabling …

Industry 4.0 technologies adoption for digital transition in drug discovery and development: a review

A Anthwal, A Uniyal, J Gairolla, R Singh… - Journal of Industrial …, 2024 - Elsevier
At present, every nation is focused on meeting sustainable development goals (SDGs) by
2030 for social, economic, and environmental sustainability. Automation of drug discovery …

[HTML][HTML] Application of artificial intelligence in modern medicine

N Xu, D Yang, K Arikawa, C Bai - Clinical eHealth, 2023 - Elsevier
Over the last decade, artificial intelligence in medicine has attracted much attention and
interest for its robust automation and efficiency in disease diagnosis, treatment and …

Pharmacological chaperones and protein conformational diseases: approaches of computational structural biology

D Grasso, S Galderisi, A Santucci, A Bernini - International Journal of …, 2023 - mdpi.com
Whenever a protein fails to fold into its native structure, a profound detrimental effect is likely
to occur, and a disease is often developed. Protein conformational disorders arise when …

Scaffold Splits Overestimate Virtual Screening Performance

Q Guo, S Hernandez-Hernandez… - … Conference on Artificial …, 2024 - Springer
Virtual Screening (VS) of vast compound libraries guided by Artificial Intelligence (AI)
models is a highly productive approach to early drug discovery. Data splitting is crucial for …

Advances in machine intelligence‐driven virtual screening approaches for big‐data

N Kumar, V Acharya - Medicinal Research Reviews, 2024 - Wiley Online Library
Virtual screening (VS) is an integral and ever‐evolving domain of drug discovery framework.
The VS is traditionally classified into ligand‐based (LB) and structure‐based (SB) …

Extended study on atomic featurization in graph neural networks for molecular property prediction

A Wojtuch, T Danel, S Podlewska… - Journal of Cheminformatics, 2023 - Springer
Graph neural networks have recently become a standard method for analyzing chemical
compounds. In the field of molecular property prediction, the emphasis is now on designing …

Analysis of metabolites in human gut: illuminating the design of gut-targeted drugs

A Gil-Pichardo, A Sánchez-Ruiz… - Journal of …, 2023 - Springer
Gut-targeted drugs provide a new drug modality besides that of oral, systemic molecules,
that could tap into the growing knowledge of gut metabolites of bacterial or host origin and …