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Recent advancements in the development of bioactive pyrazoline derivatives
Pyrazolines remain privileged heterocycles in drug discovery. 2-Pyrazoline scaffold has
been proven as a ubiquitous motif which is present in a number of pharmacologically …
been proven as a ubiquitous motif which is present in a number of pharmacologically …
[PDF][PDF] Pyrazoline derivatives: a worthy insight into the recent advances and potential pharmacological activities
MA Rahman, AA Siddiqui - Int J Pharm Sci Drug Res, 2010 - researchgate.net
Pyrazolines display a broad spectrum of potential pharmacological activities and are present
in a number of pharmacologically active molecules such as phenazone/amidopyrene …
in a number of pharmacologically active molecules such as phenazone/amidopyrene …
Synthesis, anti-bacterial and anti-fungal activities of some novel Schiff bases containing 2, 4-disubstituted thiazole ring
A series of arylidene-2-(4-(4-methoxy/bromophenyl) thiazol-2-yl) hydrazines (4a–z) and 1-(4-
(4-methoxy/bromophenyl) thiazol-2-yl)-2-cyclohexylidene/cyclopentylidene hydrazines (5a …
(4-methoxy/bromophenyl) thiazol-2-yl)-2-cyclohexylidene/cyclopentylidene hydrazines (5a …
Synthesis of new 4-thiazolidinone-, pyrazoline-, and isatin-based conjugates with promising antitumor activity
The synthesis and antitumor activity screening of novel 3-[2-(3, 5-diaryl-4, 5-dihydropyrazol-
1-yl)-4-oxo-4, 5-dihydro-1, 3-thiazol-5-ylidene]-2, 3-dihydro-1 H-indol-2-ones 1–23 and 3-(3 …
1-yl)-4-oxo-4, 5-dihydro-1, 3-thiazol-5-ylidene]-2, 3-dihydro-1 H-indol-2-ones 1–23 and 3-(3 …
Synthesis of novel thiazolone-based compounds containing pyrazoline moiety and evaluation of their anticancer activity
To examine the anticancer activity several novel thiazolone-based compounds containing 5-
aryl-3-phenyl-4, 5-dihydro-1H-pyrazol-1-yl framework were obtained. Reaction of 5-aryl-3 …
aryl-3-phenyl-4, 5-dihydro-1H-pyrazol-1-yl framework were obtained. Reaction of 5-aryl-3 …
Synthesis and antimicrobial evaluation of 1-(benzofuran-2-yl)-4-nitro-3-arylbutan-1-ones and 3-(benzofuran-2-yl)-4, 5-dihydro-5-aryl-1-[4-(aryl)-1, 3-thiazol-2-yl]-1H …
2-Acetylbenzofuran 1 on treatment with substituted aldehydes affords the corresponding
chalcones 2a–c. Treatment of the chalcones with nitromethane under Michael addition …
chalcones 2a–c. Treatment of the chalcones with nitromethane under Michael addition …
Synthesis of novel quinoline–based 4, 5–dihydro–1H–pyrazoles as potential anticancer, antifungal, antibacterial and antiprotozoal agents
A new series of N–substituted 2–pyrazolines 9a–f, 10a–f, 11a–f, 12a–f and 13a–f were
obtained from the cyclocondensation reaction of [(7–chloroquinolin–4–yl) amino] chalcones …
obtained from the cyclocondensation reaction of [(7–chloroquinolin–4–yl) amino] chalcones …
Synthesis of novel pyrazolic analogues of chalcones and their 3-aryl-4-(3-aryl-4, 5-dihydro-1H-pyrazol-5-yl)-1-phenyl-1H-pyrazole derivatives as potential antitumor …
Novel (E)-1-aryl-3-(3-aryl-1-phenyl-1H-pyrazol-4-yl) prop-2-en-1-ones 5/6 (pyrazolic
chalcones) were synthesized from a Claisen–Schmidt reaction of 3-aryl-1-phenylpyrazol-4 …
chalcones) were synthesized from a Claisen–Schmidt reaction of 3-aryl-1-phenylpyrazol-4 …
Determination of the inhibition profiles of pyrazolyl–thiazole derivatives against aldose reductase and α‐glycosidase and molecular docking studies
Aldose reductase (AR) is the first and rate‐limiting enzyme of the polyol pathway, which
converts glucose to sorbitol in an NADPH‐dependent reaction. α‐Glycosidase breaks down …
converts glucose to sorbitol in an NADPH‐dependent reaction. α‐Glycosidase breaks down …
Recent advances in the therapeutic applications of pyrazolines
Introduction: Pyrazolines are well-known and important nitrogen-containing five-membered
ring heterocyclic compounds. Various methods have been worked out for their synthesis …
ring heterocyclic compounds. Various methods have been worked out for their synthesis …