Precision Oncology: 2024 in Review

M Repetto, N Fernandez, A Drilon… - Cancer …, 2024‏ - aacrjournals.org
This article discusses the specific advances made in precision oncology in 2024. We
comment on the evolving nature of predictive molecular events used to select patients who …

Map** kinase domain resistance mechanisms for the MET receptor tyrosine kinase via deep mutational scanning

GO Estevam, E Linossi, J Rao, CB Macdonald… - eLife, 2025‏ - elifesciences.org
Mutations in the kinase and juxtamembrane domains of the MET Receptor Tyrosine Kinase
are responsible for oncogenesis in various cancers and can drive resistance to MET …

Molecular profiling METex14+ non-small cell lung cancer (NSCLC): Impact of histology

JA Marks, N Gandhi, B Halmos, ME Marmarelis… - Lung Cancer, 2024‏ - Elsevier
Objectives MET exon 14 skip** alterations (METex14+) represent a heterogeneous
subgroup of non-small cell lung cancer (NSCLC) with distinct biological and genomic …

Safety, Efficacy, and Biomarker Analysis of Crizotinib in MET-Mutated Non–Small Cell Lung Cancer—Results from the Drug Rediscovery Protocol

K Verkerk, TJWT van der Wel, LJ Zeverijn… - Clinical Cancer …, 2024‏ - aacrjournals.org
Purpose: To provide patients with MET-mutated advanced non–small cell lung cancer (MET
mut aNSCLC) access to crizotinib, further substantiate evidence of its efficacy and safety in …

[HTML][HTML] MET Exon 14 Skip** and Novel Actionable Variants: Diagnostic and Therapeutic Implications in Latin American Non-Small-Cell Lung Cancer Patients

S Rivas, RV Sepúlveda, I Tapia, C Estay… - International Journal of …, 2024‏ - mdpi.com
Targeted therapy indications for actionable variants in non-small-cell lung cancer (NSCLC)
have primarily been studied in Caucasian populations, with limited data on Latin American …

Prospective evaluation of structure-based simulations reveal their ability to predict the impact of kinase mutations on inhibitor binding

S Singh, V Gapsys, M Aldeghi, D Schaller… - bioRxiv, 2024‏ - biorxiv.org
Small molecule kinase inhibitors are critical in the modern treatment of cancers, evidenced
by the existence of over 80 FDA-approved small-molecule kinase inhibitors. Unfortunately …

Response to Crizotinib After Entrectinib Resistance in ROS1-Rearranged, MET-Amplified Lung Adenocarcinoma

VR Vaz, MM Gandhi, B Ricciuti, JV Alessi… - JCO Precision …, 2024‏ - ascopubs.org
Response to Crizotinib After Entrectinib Resistance in ROS1-Rearranged, MET-Amplified Lung
Adenocarcinoma | JCO Precision Oncology Skip to main content ASCO Publications …

[PDF][PDF] MET Exon 14 Skip** and Novel Actionable Variants: Diagnostic and Therapeutic Implications in Latin American NSCLC patients.

S Rivas, RV Sepulveda, I Tapia, C Estay, V Soto… - 2024‏ - preprints.org
Targeted therapy indications for actionable variants in non-small cell lung cancer (NSCLC)
have primarily been studied in Caucasian populations, with limited data on Latin American …

Resistance to Allosteric Inhibitors

I Outhwaite, I Kwan, NP Shah, I Bahar… - Available at SSRN …‏ - papers.ssrn.com
Allosteric inhibitors have emerged as powerful therapeutic agents capable of overcoming
resistance mutations that impair the efficacy of orthosteric inhibitors. However, resistance to …