Pd-Catalyzed Intermolecular ortho-C−H Amidation of Anilides by N-Nosyloxycarbamate

KH Ng, ASC Chan, WY Yu - Journal of the American Chemical …, 2010 - ACS Publications
A palladium-catalyzed ortho-C− H amidation of anilides by N-nosyloxycarbamates was
developed for the synthesis of 2-aminoanilines. This reaction can be carried out under …

Recent advances of bismuth (III) salts in organic chemistry: application to the synthesis of heterocycles of pharmaceutical interest

JAR Salvador, R Pinto… - Current Organic Synthesis, 2009 - ingentaconnect.com
The use of bismuth (III) salts in organic synthesis has attracted an increasing interest over
the last years. Systems comprising of bismuth (III) salts are generally catalytic and involve a …

Nonpeptidic ligands for peptide-activated G protein-coupled receptors

JS Blakeney, RC Reid, GT Le, DP Fairlie - Chemical reviews, 2007 - ACS Publications
There are some 850 human G protein-coupled receptors (GPCRs) currently known
(http://bioinformatics2. biol. uoa. gr), making this the most abundant family of well …

Discovery of tetrazolamide-benzimidazol-2-ones as novel 4-Hydroxyphenylpyruvate dioxygenase inhibitors

ZM Cai, GY Huang, J Dong, LJ Chen… - Journal of Agricultural …, 2024 - ACS Publications
4-Hydroxyphenylpyruvate dioxygenase (HPPD, EC 1.13. 11.27) is one of the most valuable
herbicide targets due to its unique biological functions. In search of HPPD inhibitors with …

Synthesis and biological evaluation of analogues of AKT (protein kinase B) inhibitor-IV

Q Sun, R Wu, S Cai, Y Lin, L Sellers… - Journal of medicinal …, 2011 - ACS Publications
Inhibitors of the PI3-kinase/AKT (protein kinase B) pathway are under investigation as
anticancer and antiviral agents. The benzimidazole derivative AKT inhibitor-IV (ChemBridge …

Desulfurization mediated by hypervalent iodine (III): A novel strategy for the construction of heterocycles

H Ghosh, R Yella, J Nath, BK Patel - 2008 - Wiley Online Library
The desulfurization ability of diacetoxyiodobenzene (DIB) has been explored in the
preparation of isothiocyanates from the corresponding dithiocarbamate salts. The in situ …

[Cp* RhCl 2] 2-catalyzed ortho-C–H bond amination of acetophenone o-methyloximes with primary N-chloroalkylamines: convenient synthesis of N-alkyl-2 …

KH Ng, Z Zhou, WY Yu - Chemical Communications, 2013 - pubs.rsc.org
Rh (III)-catalyzed aromatic C–H amination of acetophenone o-methyloximes with primary N-
chloroalkylamines was developed, and the arylamine products were obtained in up to 92 …

[HTML][HTML] An effective microwave-induced iodine-catalyzed method for the synthesis of quinoxalines via condensation of 1, 2-diamines with 1, 2-dicarbonyl compounds

D Bandyopadhyay, S Mukherjee, RR Rodriguez… - Molecules, 2010 - mdpi.com
Molecules | Free Full-Text | An Effective Microwave-Induced Iodine-Catalyzed Method for the
Synthesis of Quinoxalines via Condensation of 1,2-Diamines with 1,2-Dicarbonyl Compounds …

Benzimidazole derivatives as tubulin polymerization inhibitors: design, synthesis and in vitro cytotoxicity studies

K Laxmikeshav, Z Rahman, A Mahale… - Bioorganic & Medicinal …, 2023 - Elsevier
A new class of benzimidazole derivatives as tubulin polymerization inhibitors has been
designed and synthesized in this study. The in vitro anticancer profile of the developed …

Benzimidazole based bis-carboxamide derivatives as promising cytotoxic agents: Design, synthesis, in silico and tubulin polymerization inhibition

K Laxmikeshav, P Sharma, M Palepu, P Sharma… - Journal of Molecular …, 2023 - Elsevier
A new series of carboxamide-bearing benzimidazole derivatives have been reported for
their cytotoxicity profile (in vitro) on selected human tumour cells like A549, HCT116, SK-Mel …