Structure–function relationships in aryl diazirines reveal optimal design features to maximize C–H insertion

SF Musolino, Z Pei, L Bi, GA DiLabio, JE Wulff - Chemical Science, 2021 - pubs.rsc.org
Diazirine reagents allow for the ready generation of carbenes upon photochemical, thermal,
or electrical stimulation. Because carbenes formed in this way can undergo rapid insertion …

Efficient synthesis of photoreactive 2-propoxyaniline derivatives as artificial sweeteners

Y Murai, T Yoshida, L Wang, K Masuda, Y Hashidoko… - Synlett, 2016 - thieme-connect.com
5-Nitro-2-propoxyaniline is one of the strongest artificial sweeteners. However, little is known
about the detailed relationship of the structure and biological activity between 5-nitro-2 …

Asymmetric synthesis of photophore-containing lactisole derivatives to elucidate sweet taste receptors

T Nakagita, A Ishida, ZP Tachrim, L Wang, T Misaka… - Molecules, 2020 - mdpi.com
Lactisole, which has a 2-phenoxy propionic acid skeleton, is well-known as an inhibitor of
sweet taste receptors. We recently revealed some of the structure–activity relationships of …

Efficient upcycling of low-functionality polymers using trifluoromethyl aryl diazirine chemistry

L Bi - 2023 - dspace.library.uvic.ca
Crosslinking technologies are widely employed in our daily life: from silicone bakeware to
epoxy adhesives and rubber tires. Traditionally, however, each type of commodity polymer …

[PDF][PDF] Synthesis of benzophenone and phenylazide derivatives of salicin for functional analysis of the bitter taste receptor using photoaffinity labeling

T Yoshida, Y Hashidoko, M Hashimoto - Heterocycles, 2016 - triggered.edina.clockss.org
Salicin is a substance that is well known for its bitter taste. Photoreactive benzophenone and
phenylazide derivatives of salicin are for the functional analysis of interactions between the …

[PDF][PDF] A New Antiplasmodial Compound from the Papuan Marine Sponge Xestospongia sp.

U Supratman - 2018 - academia.edu
Abstract A new antiplasmodial compound, 2-(3H-diazirine-3-yl) benzaldehyde (1), has been
isolated from the Papuan marine sponge Xestospongia sp. The structure elucidation of …

[CITATION][C] A new antiplasmodial compound from the Papuan marine sponge Xestospongia sp

AMS Murtihapsari, DK Kadarusman… - 2018 - UIN Syarif Hidayatullah, Jakarta