Molecular docking: a powerful approach for structure-based drug discovery

XY Meng, HX Zhang, M Mezei… - Current computer-aided …, 2011‏ - ingentaconnect.com
Molecular docking has become an increasingly important tool for drug discovery. In this
review, we present a brief introduction of the available molecular docking methods, and their …

Relevance of molecular docking studies in drug designing

R Jakhar, M Dangi, A Khichi… - Current …, 2020‏ - benthamdirect.com
Molecular Docking is used to positioning the computer-generated 3D structure of small
ligands into a receptor structure in a variety of orientations, conformations and positions …

Molecular similarity: a key technique in molecular informatics

A Bender, RC Glen - Organic & biomolecular chemistry, 2004‏ - pubs.rsc.org
Molecular Informatics utilises many ideas and concepts to find relationships between
molecules. The concept of similarity, where molecules may be grouped according to their …

Deep learning in structural bioinformatics: current applications and future perspectives

N Kumar, R Srivastava - Briefings in Bioinformatics, 2024‏ - academic.oup.com
In this review article, we explore the transformative impact of deep learning (DL) on
structural bioinformatics, emphasizing its pivotal role in a scientific revolution driven by …

Insights into the mode of inhibition of human mitochondrial monoamine oxidase B from high-resolution crystal structures

C Binda, M Li, F Hubálek, N Restelli… - Proceedings of the …, 2003‏ - pnas.org
Monoamine oxidase B (MAO-B) is an outer mitochondrial membrane-bound enzyme that
catalyzes the oxidative deamination of arylalkylamine neurotransmitters and has been a …

Recent progress in development of dopamine receptor subtype-selective agents: potential therapeutics for neurological and psychiatric disorders

A Zhang, JL Neumeyer, RJ Baldessarini - Chemical reviews, 2007‏ - ACS Publications
Dopamine (DA) is a critical neurotransmitter in the mammalian central nervous system
(CNS). The cerebral dopaminergic system is implicated in the pathophysiology of several …

Protein flexibility and drug design: how to hit a moving target

HA Carlson - Current opinion in chemical biology, 2002‏ - Elsevier
The most advanced methods for computer-aided drug design and database mining
incorporate protein flexibility. Such techniques are not only needed to obtain proper results; …

Computational approaches to identifying and characterizing protein binding sites for ligand design

S Henrich, OMH Salo‐Ahen, B Huang… - Journal of Molecular …, 2010‏ - Wiley Online Library
Given the three‐dimensional structure of a protein, how can one find the sites where other
molecules might bind to it? Do these sites have the properties necessary for high affinity …

Protein flexibility in docking and surface map**

KW Lexa, HA Carlson - Quarterly reviews of biophysics, 2012‏ - cambridge.org
Structure-based drug design has become an essential tool for rapid lead discovery and
optimization. As available structural information has increased, researchers have become …

Chemometrics

B Lavine, J Workman - Analytical chemistry, 2008‏ - ACS Publications
This review, the seventeenth of this series and the fifteenth with the title of Chemometrics,
covers the most significant developments in the field from January 2006 through December …