Molecular biomarkers in acute myeloid leukemia

J Prada-Arismendy, JC Arroyave, S Röthlisberger - Blood reviews, 2017 - Elsevier
Acute myeloid leukemia (AML) is the most common acute leukemia in adults. The
pathophysiology of this disease is just beginning to be understood at the cellular and …

Pharmacological inhibition of LSD1 for cancer treatment

GJ Yang, PM Lei, SY Wong, DL Ma, CH Leung - Molecules, 2018 - mdpi.com
Lysine-specific demethylase 1A (LSD1, also named KDM1A) is a demethylase that can
remove methyl groups from histones H3K4me1/2 and H3K9me1/2. It is aberrantly expressed …

[HTML][HTML] TP53 and Decitabine in Acute Myeloid Leukemia and Myelodysplastic Syndromes

JS Welch, AA Petti, CA Miller, CC Fronick… - … England Journal of …, 2016 - Mass Medical Soc
Background The molecular determinants of clinical responses to decitabine therapy in
patients with acute myeloid leukemia (AML) or myelodysplastic syndromes (MDS) are …

A comprehensive review of lysine-specific demethylase 1 and its roles in cancer

A Hosseini, S Minucci - Epigenomics, 2017 - Taylor & Francis
Histone methylation plays a key role in the regulation of chromatin structure, and its
dynamics regulates important cellular processes. The investigation of the role of alterations …

Therapeutic potential of targeting LSD1/KDM1A in cancers

X Zhang, X Wang, T Wu, W Yin, J Yan, Y Sun… - Pharmacological …, 2022 - Elsevier
LSD1 was the first histone demethylase identified by Professor Shi Yang and his team
members in 2004. LSD1 employs FAD as its cofactor, which catalyzes the demethylation of …

IGF2 is up-regulated by epigenetic mechanisms in hepatocellular carcinomas and is an actionable oncogene product in experimental models

I Martinez-Quetglas, R Pinyol, D Dauch, S Torrecilla… - Gastroenterology, 2016 - Elsevier
Background & Aims Effective treatments are urgently needed for hepatocellular carcinoma
(HCC), which is usually diagnosed at advanced stages. Signaling via the insulin-like growth …

Roles and epigenetic regulation of epithelial–mesenchymal transition and its transcription factors in cancer initiation and progression

JY Lee, G Kong - Cellular and molecular life sciences, 2016 - Springer
The epithelial–mesenchymal transition (EMT) is a crucial developmental process by which
epithelial cells undergo a mesenchymal phenotypic change. During EMT, epigenetic …

The genetic and molecular pathogenesis of myelodysplastic syndromes

RM Shallis, R Ahmad, AM Zeidan - European journal of …, 2018 - Wiley Online Library
Myelodysplastic syndromes (MDS) comprise a diverse group of clonal and malignant
myeloid disorders characterized by ineffective hematopoiesis, resultant peripheral …

N6-Adenosine Methylation (m6A) RNA Modification: an Emerging Role in Cardiovascular Diseases

Y Chen, X Ouyang, X Yu, P Novák, L Zhou… - Journal of …, 2021 - Springer
Abstract N6-methyladenosine (m 6 A) is the most abundant and prevalent epigenetic
modification of mRNA in mammals. This dynamic modification is regulated by m 6 A …

Epigenetics in cancer: a hematological perspective

M Stahl, N Kohrman, SD Gore, TK Kim, AM Zeidan… - PLoS …, 2016 - journals.plos.org
For several decades, we have known that epigenetic regulation is disrupted in cancer.
Recently, an increasing body of data suggests epigenetics might be an intersection of …