Isoxazoles and their derivatives represent privileged heteroaromatic motifs, which exhibit
remarkable biological and pharmaceutical activities. Notably, metal catalyzed or mediated …

Isoxazole derivatives are aromatic five-membered ring heterocyclic compounds with one
oxygen atom and one nitrogen atom at adjacent positions. These compounds have a broad …

The cross-coupling reaction of 1, 3, 5-triethynylbenzene with terephthaloyl chloride gives a
novel ynone-linked porous organic polymer. Tethering alkyl amine species on the polymer …

Herein, we report a Pd‐catalyzed enantioselective domino Heck carbonylation reaction of o‐
iodoacrylanilides with terminal alkynes and water as the nucleophiles, affording a diversity …

In this study, 56 isoxazole derivatives were synthesized and their antitumor activity against 9
cancer cells, such as BXPC-3, MiaPaCa-2, PANC-1, MCF-7, HCT-116, HepG2, NCI-H460 …

Isoxazol (in) es are widely featured structural motifs in natural products, agrochemicals, and
pharmaceuticals. The first intermolecular approach for a direct electrochemical synthesis …

A facile synthetic route toward either 3-or 5-fluoroalkyl-substituted isoxazoles or pyrazoles
containing an additional functionalization site was developed and applied on a multigram …

A general method for the synthesis of isoselenazoles and isothiazoles has been developed
by the base-promoted demethoxylative cycloaddition of alkynyl oxime ethers using the …

Various primary alcohols were smoothly transformed into 3-aryl-and 3-alkylisoxazoles in
good yields in one pot by successive treatment with PhI (OAc) 2 in the presence of TEMPO …

An efficient synthesis of bisisothiazole-4-yl disulfides via the demethoxylative thioannulation
of alkynyl oxime ethers with odorless elemental sulfur has been first developed. This …