[HTML][HTML] Synthesis of ethyl pyrimidine-quinolincarboxylates selected from virtual screening as enhanced lactate dehydrogenase (LDH) inhibitors

I Díaz, S Salido, M Nogueras, J Cobo - International Journal of Molecular …, 2024 - mdpi.com
The inhibition of the hLDHA (human lactate dehydrogenase A) enzyme has been
demonstrated to be of great importance in the treatment of cancer and other diseases, such …

[HTML][HTML] Qualitative Profiling, Antioxidant and Antimicrobial Activities of Polar and Nonpolar Basil Extracts

V Vidaković, B Vujić, M Jadranin, I Novaković… - Foods, 2024 - mdpi.com
Basil (Ocimum basilicum L.) is a widely used culinary herb. In this study, ethanol,
dichloromethane, and sunflower oil were used separately as solvents with distinct polarities …

Discovery of a new class of potent pyrrolo [3, 4-c] quinoline-1, 3-diones based inhibitors of human dihydroorotate dehydrogenase: Synthesis, pharmacological and …

MG Dimitrijević, C Roschger, K Lang, A Zierer… - Bioorganic …, 2024 - Elsevier
Abstract Twenty N-substituted pyrrolo [3, 4-c] quinoline-1, 3-diones 3a-t were synthesized by
a cyclization reaction of Pfitzinger's quinoline ester precursor with the selected aromatic …

Discovery a series of novel inhibitors of human dihydroorotate dehydrogenase: Biological activity evaluation and molecular docking

X Ren, X Liu, M Hua, Y Dai, X Ren… - Chemical Biology & …, 2024 - Wiley Online Library
Human dihydroorotate dehydrogenase (h DHODH) is a key enzyme that catalyzes the de
novo synthesis of pyrimidine. In recent years, various studies have shown that inhibiting this …