Nitrogen containing heterocycles as anticancer agents: A medicinal chemistry perspective

A Kumar, AK Singh, H Singh, V Vijayan, D Kumar… - Pharmaceuticals, 2023‏ - mdpi.com
Cancer is one of the major healthcare challenges across the globe. Several anticancer
drugs are available on the market but they either lack specificity or have poor safety, severe …

Prescribed drugs containing nitrogen heterocycles: an overview

MM Heravi, V Zadsirjan - RSC advances, 2020‏ - pubs.rsc.org
Heteroatoms as well as heterocyclic scaffolds are frequently present as the common cores in
a plethora of active pharmaceuticals natural products. Statistically, more than 85% of all …

A review on recent advances in nitrogen-containing molecules and their biological applications

N Kerru, L Gummidi, S Maddila, KK Gangu… - Molecules, 2020‏ - mdpi.com
The analogs of nitrogen-based heterocycles occupy an exclusive position as a valuable
source of therapeutic agents in medicinal chemistry. More than 75% of drugs approved by …

Recent advances in chemistry and therapeutic potential of functionalized quinoline motifs–a review

OO Ajani, KT Iyaye, OT Ademosun - RSC advances, 2022‏ - pubs.rsc.org
Quinoline, which consists of benzene fused with N-heterocyclic pyridine, has received
considerable attention as a core template in drug design because of its broad spectrum of …

[HTML][HTML] Novel pyridine and pyrimidine derivatives as promising anticancer agents: A review

M Albratty, HA Alhazmi - Arabian Journal of Chemistry, 2022‏ - Elsevier
Pyridines and pyrimidines are the class of heterocyclic nitrogenous compounds having
plethora of applications in anticancer drug development. These synthetic sources serve as …

Bioactive pyrrole-based compounds with target selectivity

GL Petri, V Spano, R Spatola, R Holl… - European journal of …, 2020‏ - Elsevier
The discovery of novel synthetic compounds with drug-like properties is an ongoing
challenge in medicinal chemistry. Natural products have inspired the synthesis of …

Natural source, bioactivity and synthesis of benzofuran derivatives

Y Miao, Y Hu, J Yang, T Liu, J Sun, X Wang - RSC advances, 2019‏ - pubs.rsc.org
Benzofuran compounds are a class of compounds that are ubiquitous in nature. Numerous
studies have shown that most benzofuran compounds have strong biological activities such …

Pharmacological significance of nitrogen-containing five and six-membered heterocyclic scaffolds as potent cholinesterase inhibitors for drug discovery

RJ Obaid, EU Mughal, N Naeem, MM Al-Rooqi… - Process …, 2022‏ - Elsevier
N-heterocycles are crucial due to their biological, chemical, and practical significance. They
are heavily investigated in biological processes involving anticancer, anti-inflammatory …

Hepatocellular carcinoma: etiology and current and future drugs

A **dal, A Thadi, K Shailubhai - Journal of clinical and experimental …, 2019‏ - Elsevier
Hepatocellular carcinoma (HCC) is swiftly increasing in prevalence globally with a high
mortality rate. The progression of HCC in patients is induced with advanced fibrosis, mainly …

Comprehensive review on the Bis–heterocyclic compounds and their anticancer efficacy

MHA Al-Jumaili, AA Hamad, HE Hashem… - Journal of Molecular …, 2023‏ - Elsevier
Heterocyclic compounds are one of the largest family of organic compounds with broad
range of applications in medicinal chemistry and agrochemicals product. Bis-heterocycle …