Machine learning in preclinical drug discovery

DB Catacutan, J Alexander, A Arnold… - Nature Chemical …, 2024‏ - nature.com
Drug-discovery and drug-development endeavors are laborious, costly and time consuming.
These programs can take upward of 12 years and cost US $2.5 billion, with a failure rate of …

Unlocking the potential of generative AI in drug discovery

A Gangwal, A Lavecchia - Drug Discovery Today, 2024‏ - Elsevier
Highlights•Artificial intelligence (AI) is transforming the drug discovery process by providing
actionable insights from huge amount of data.•Deep-learning models, especially generative …

Current strategies to address data scarcity in artificial intelligence-based drug discovery: A comprehensive review

A Gangwal, A Ansari, I Ahmad, AK Azad… - Computers in Biology …, 2024‏ - Elsevier
Artificial intelligence (AI) has played a vital role in computer-aided drug design (CADD). This
development has been further accelerated with the increasing use of machine learning (ML) …

Tackling assay interference associated with small molecules

L Tan, S Hirte, V Palmacci, C Stork… - Nature Reviews …, 2024‏ - nature.com
Biochemical and cell-based assays are essential to discovering and optimizing efficacious
and safe drugs, agrochemicals and cosmetics. However, false assay readouts stemming …

Industry-scale orchestrated federated learning for drug discovery

M Oldenhof, G Ács, B Pejó, A Schuffenhauer… - Proceedings of the aaai …, 2023‏ - ojs.aaai.org
To apply federated learning to drug discovery we developed a novel platform in the context
of European Innovative Medicines Initiative (IMI) project MELLODDY (grant n 831472) …

Deep learning models compared to experimental variability for the prediction of CYP3A4 time-dependent inhibition

A Fluetsch, M Trunzer, G Gerebtzoff… - Chemical research in …, 2024‏ - ACS Publications
Most drugs are mainly metabolized by cytochrome P450 (CYP450), which can lead to drug–
drug interactions (DDI). Specifically, time-dependent inhibition (TDI) of CYP3A4 isoenzyme …

Recent advances in generative biology for biotherapeutic discovery

M Mock, CJ Langmead, P Grandsard… - Trends in …, 2024‏ - cell.com
Generative biology combines artificial intelligence (AI), advanced life sciences technologies,
and automation to revolutionize the process of designing novel biomolecules with …

Prediction of Small-Molecule Developability Using Large-Scale In Silico ADMET Models

M Beckers, N Sturm, F Sirockin… - Journal of medicinal …, 2023‏ - ACS Publications
Early in silico assessment of the potential of a series of compounds to deliver a drug is one
of the major challenges in computer-assisted drug design. The goal is to identify the right …

Multi-party collaborative drug discovery via federated learning

D Huang, X Ye, T Sakurai - Computers in Biology and Medicine, 2024‏ - Elsevier
In the field of drug discovery and pharmacology research, precise and rapid prediction of
drug-target binding affinity (DTA) and drug-drug interaction (DDI) are essential for drug …

Another string to your bow: Machine learning prediction of the pharmacokinetic properties of small molecules

D Bassani, NJ Parrott, N Manevski… - Expert Opinion on Drug …, 2024‏ - Taylor & Francis
Introduction Prediction of pharmacokinetic (PK) properties is crucial for drug discovery and
development. Machine-learning (ML) models, which use statistical pattern recognition to …