Inhibition of monoamine oxidase by selected C5-and C6-substituted isatin analogues

CI Manley-King, JJ Bergh, JP Petzer - Bioorganic & medicinal chemistry, 2011 - Elsevier
Previous studies have shown that (E)-5-styrylisatin and (E)-6-styrylisatin are reversible
inhibitors of human monoamine oxidase (MAO) A and B. Both homologues are reported to …

Inhibition of monoamine oxidase by 8-benzyloxycaffeine analogues

B Strydom, SF Malan, N Castagnoli Jr, JJ Bergh… - Bioorganic & medicinal …, 2010 - Elsevier
Based on recent reports that several (E)-8-styrylcaffeinyl analogues are potent reversible
inhibitors of monoamine oxidase B (MAO-B), a series of 8-benzyloxycaffeinyl analogues …

Reactivity and kinetics of vinyl sulfone-functionalized self-assembled monolayers for bioactive ligand immobilization

H Wang, F Cheng, M Li, W Peng, J Qu - Langmuir, 2015 - ACS Publications
A new vinyl sulfone (VS) disulfide, 1, 2-bis (11-(vinyl sulfonyl) undecyl) disulfane, was
synthesized to enable the preparation of VS-presenting self-assembled monolayers (VS …

A challenging Heck reaction of maleimides

LH Lim, JS Zhou - Organic Chemistry Frontiers, 2015 - pubs.rsc.org
A challenging Heck reaction of maleimides - Organic Chemistry Frontiers (RSC Publishing)
DOI:10.1039/C5QO00015G Royal Society of Chemistry View PDF VersionPrevious ArticleNext …

8-Aryl-and alkyloxycaffeine analogues as inhibitors of monoamine oxidase

B Strydom, JJ Bergh, JP Petzer - European journal of medicinal chemistry, 2011 - Elsevier
Recently it was reported that a series of 8-benzyloxycaffeine analogues are potent
reversible inhibitors of human monoamine oxidase (MAO) A and B. In an attempt to discover …

HFIP-promoted Michael reactions: direct para-selective C–H activation of anilines with maleimides

B Li, Q Mao, J Zhou, F Liu, N Ye - Organic & Biomolecular Chemistry, 2019 - pubs.rsc.org
The Michael reaction is widely used for the C–C coupling of electron-poor olefins and C
(sp3)–H pronucleophiles. Herein, an effective Michael reaction approach between electron …

Single Heterocyclic Compounds as Monoamine Oxidase Inhibitors: From Past to Present

SM Wu, XY Qiu, SJ Liu, J Sun - Mini Reviews in Medicinal …, 2020 - ingentaconnect.com
Inhibitors of monoamine oxidase (MAO) have shown therapeutic values in a variety of
neurodegenerative diseases such as depression, Parkinson's disease and Alzheimer's …

Selective and tunable synthesis of 3-arylsuccinimides and 3-arylmaleimides from arenediazonium tetrafluoroborates and maleimides

ZH Yang, ZH Chen, YL An, SY Zhao - RSC advances, 2016 - pubs.rsc.org
A highly efficient synthetic strategy for synthesizing 3-arylsuccinimides has been developed
from arenediazonium tetrafluoroborates and maleimides in the presence of TiCl3. The …

Visible-light-promoted Meerwein 3, 4-diarylation of maleimides with electron-deficient diazonium salts

AD Kharlamova, AS Abel, VE Gontcharenko, AD Averin… - Tetrahedron, 2024 - Elsevier
Diarylmaleimides are widely explored as structural fragments of natural products, bioactive
substances and components of luminescent materials. The reaction of aryl diazonium salts …

Palladium‐Catalyzed Carbonylative Cyclization of Terminal Alkynes and Anilines to 3‐Substituted Maleimides

JX Xu, XF Wu - Advanced Synthesis & Catalysis, 2018 - Wiley Online Library
Herein, we describe an interesting palladium‐catalyzed protocol for the carbonylative
synthesis of 3‐substituted maleimides. By annulation of simple anilines with terminal …