1, 3, 4‐Thiadiazole and its derivatives: A review on recent progress in biological activities

AK Jain, S Sharma, A Vaidya… - Chemical biology & …, 2013 - Wiley Online Library
The 1, 3, 4‐thiadiazole nucleus is one of the most important and well‐known heterocyclic
nuclei, which is a common and integral feature of a variety of natural products and medicinal …

[HTML][HTML] Synthesis, characterization and antimicrobial activity of peanut skin extract-azo-compounds

SK Kyei, O Akaranta, G Darko - Scientific African, 2020 - Elsevier
Peanut skin extract, an agro-waste and a source of flavonoids has been extracted from
peanut skin and employed as a precursor for the synthesis of novel azo compounds and …

Design, synthesis, and characterization of a novel pH-responsive azo dye incorporating a 1, 3, 4-thiadiazole ring for advanced textile applications

S Belowar, M Rahamatolla, S Islam, MA Jalil… - Dyes and …, 2024 - Elsevier
This study presents the synthesis and comprehensive characterization of a novel azo dye
derived from 2-(5-amino-1, 3, 4-thiadiazol-2-yl) phenol (1a). The synthesis was initiated by …

1, 3, 4-Thiadiazole-containing azo dyes: Synthesis, spectroscopic properties and molecular structure

A Kudelko, M Olesiejuk, M Luczynski, M Swiatkowski… - Molecules, 2020 - mdpi.com
Three series of azo dyes derived from 2-amino-5-aryl-1, 3, 4-thiadiazoles and aniline, N, N-
dimethylaniline and phenol were synthesized in high yields by a conventional diazotization …

[HTML][HTML] Synthesis, characterization and comparative study the microbial activity of some heterocyclic compounds containing oxazole and benzothiazole moieties

IHR Tomi, JH Tomma, AHR Al-Daraji… - Journal of Saudi Chemical …, 2015 - Elsevier
New derivatives of five member heterocyclic compounds containing oxazole and
benzothiazole rings are reported. These compounds have been characterized by elemental …

Synthesis and evaluation of novel 1, 3, 4-thiadiazole--fluoroquinolone hybrids as antibacterial, antituberculosis, and anticancer agents

A Demirci, KG KARAYEL, E Tatar… - Turkish Journal of …, 2018 - journals.tubitak.gov.tr
Abstract A series of 5-substituted-1, 3, 4-thiadiazole-based fluoroquinolone derivatives were
designed as potential antibacterial and anticancer agents using a molecular hybridization …

[HTML][HTML] Synthesis, antimicrobial and docking study of three novel 2, 4, 5-triarylimidazole derivatives

IHR Tomi, AHR Al-Daraji, AM Abdula… - Journal of Saudi …, 2016 - Elsevier
Abstract A novel series of 2-[5-(4-substituted phenyl) furan-2-yl]-4, 5-diphenyl-1H-imidazole
derivatives (2a–c) were synthesized and characterized using IR, 1 H NMR and GC–MS …

Design, synthesis, spectral characterization and molecular docking studies of novel pyranoquinolinyl dihydropyridine carboxylates as potential antibacterial agents …

G Lavanya, CJ Magesh, K Venkatapathy… - Bioorganic …, 2021 - Elsevier
Novel pyranoquinolinyl dihydropyridine carboxylate (PDC) derivatives were designed by
incorporating the multi-drug resistance modulating effects of 1, 4 dihydropyridines along with …

Microwave-Assisted Facile Synthesis, Anticancer Evaluation and Docking Study of N-((5-(Substituted methylene amino)-1,3,4-thiadiazol-2-yl)methyl) Benzamide …

SV Tiwari, S Siddiqui, JA Seijas, MP Vazquez-Tato… - Molecules, 2017 - mdpi.com
In the present work, 12 novel Schiff's bases containing a thiadiazole scaffold and benzamide
groups coupled through appropriate pharmacophore were synthesized. These moieties are …

[PDF][PDF] Synthesis, docking study and in vitro anticancer evaluation of new derivatives of 2-(1-(2-flouro-[1, 1-biphenyl]-4-yl) ethyl)-6-(substituted phenyl) imidazole [2, 1-B …

KS Hmood, AARM Kubba - Systematic Reviews in Pharmacy, 2020 - academia.edu
Results: The new compounds were characterized by FTIR, 1HNMRs and CHNS analysis. A
molecular docking study of the synthesized compounds (2-5) against HIV protease indicated …