Solid-phase synthesis of quinolinone library

S Kwak, MJ Kim, SD Lee, H You… - ACS Combinatorial …, 2015 - ACS Publications
Quinolinones have various biological activities, including antibacterial, anticancer, and
antiviral properties. The 3-substituted amide quinolin-2 (1 H)-ones not only show …

Polymorphism and the analgesic activity of N-(3-pyridylmethyl)-4-hydroxy-2-oxo-1, 2, 5, 6, 7, 8-hexahydroquinoline-3-carboxamide

IV Ukrainets, OV Mospanova… - Journal of Organic …, 2015 - ophcj.nuph.edu.ua
The advanced study of the analgesic activity of N-(3-pyridylmethyl)-4-hydroxy-2-oxo-1, 2, 5,
6, 7, 8-hexahydroquinoline-3-carboxamide selected by the results of the primary …

[PDF][PDF] Synthesis of 2-oxoquinoline-3-carboxamide of ampicillin and amoxicillin as inhibitors of penicillin binding protein 1A of Pseudomonas aeruginosa

J Shelke, G Meshram, P Dongre - Acta Poloniae Pharmaceutica-Drug …, 2012 - ptfarm.pl
A series of ampicillin and amoxicillin derivatives were prepared by N-acylation with N1-
substituted 1, 2-dihydro-2-oxoquinoline carboxylic acids by Schotten-Baumann procedure …

Synthesis and diuretic properties of N-aryl-6-hydroxy-2-methyl-4-oxo-2, 4-dihydro-1H-pyrrolo [3, 2, 1-ij] quinoline-5-carboxamides with electron-acceptor substituents …

IV Ukrainets, MY Golik, OL Shemchuk, VM Kravchenko - 2013 - dspace.nuph.edu.ua
In numerous studies of 4-hydroxy-2-oxo-1, 2-dihydroquinoline-3-carboxamides it has been
convincingly shown that amidation of quinoline-3-carboxylic acids esters with alkyl-, aryl-and …

2-Acylcycloalkanones in Organic Synthesis

VD Dyachenko, SM Sukach, AS Morkovnik - Russian Journal of Organic …, 2020 - Springer
2-Acylcycloalkanones in Organic Synthesis | Russian Journal of Organic Chemistry Skip to
main content SpringerLink Account Menu Find a journal Publish with us Track your …

Синтез, строение и противотуберкулезная активность NR-амидов 4-гидрокси-1-изо-бутил-2-оксо-1, 2, 5, 6, 7, 8-гексагидрохинолин-3-карбоновой кислоты

ИВ Украинец, ЕВ Моспанова… - Журнал органічної …, 2011 - dspace.nbuv.gov.ua
На примере анилидов и гетариламидов 4-гидрокси-1-изо-бутил-2-оксо-1, 2, 5, 6, 7, 8-
гексагидрохинолин-3-карбоновой кислоты показано, что на противотуберкулезные …

[PDF][PDF] Створення нових діуретиків на основі похідних хінолону-2

МЮ Голік - 2021 - dspace.nuph.edu.ua
Національний фармацевтичний університет Міністерство охорони здоро Page 1
Національний фармацевтичний університет Міністерство охорони здоров’я України …

The synthesis and the antitubercular activity of 1-benzyl-4-hydroxy-2-oxo-1, 2, 5, 6, 7, 8-hexahydroquinoline-3-carboxamides

OO Davydenko - Journal of Organic and Pharmaceutical …, 2015 - ophcj.nuph.edu.ua
Unfortunately, tuberculosis still remains a cause of high mortality in humans and in modern
conditions it has become a global health problem. Continuing the search for new …

Synthesis and diuretic properties of N-aryl-6-hydroxy-2-methyl-4-oxo-2, 4-dihydro-1H-pyrrolo

IV Ukrainets, MY Golik, OL Shemchuk… - Журнал органічної …, 2013 - irbis-nbuv.gov.ua
In numerous studies of 4-hydroxy-2-oxo-1, 2-dihydroquinoline-3-carboxamides it has been
convincingly shown that amidation of quinoline-3-carboxylic acids esters with alkyl-, aryl-and …

Studium kondenzace N-substituovaných cyklických iminů s malonáty

L Tatarková - 2018 - digilib.k.utb.cz
Předmětem teoretické části v předložené bakalářské práci se staly deriváty 4-hydroxypyridin-
2 (1H)-onu a 4-hydroxychinolin-2 (1H)-onu, a to jak po stránce biologické aktivy, tak i po …