Fluorescent Probes and Quenchers in Studies of Protein Folding and Protein‐Lipid Interactions

A Kyrychenko, AS Ladokhin - The Chemical Record, 2024‏ - Wiley Online Library
Fluorescence spectroscopy provides numerous methodological tools for structural and
functional studies of biological macromolecules and their complexes. All fluorescence …

Opportunities and challenges of fatty acid conjugated therapeutics

M Bhat, R Jatyan, A Mittal, RI Mahato… - Chemistry and Physics of …, 2021‏ - Elsevier
Instability, poor cellular uptake and unfavorable pharmacokinetics and biodistribution of
many therapeutic molecules require modification in their physicochemical properties. The …

From haemadin to haemanorm: Synthesis and characterization of full‐length haemadin from the leech Haemadipsa sylvestris and of a novel bivalent, highly potent …

L Acquasaliente, A Pierangelini, A Pagotto… - Protein …, 2023‏ - Wiley Online Library
Hirudin from Hirudo medicinalis is a bivalent α‐Thrombin (αT) inhibitor, targeting the enzyme
active site and exosite‐I, and is currently used in anticoagulant therapy along with its …

Indolizinylalanine Regioisomers: Tryptophan Isosteres with Bathochromic Fluorescence Emission

GID Cooper, I Saha, J Newman, RH Shin… - The Journal of …, 2024‏ - ACS Publications
We have developed a high yielding synthesis of indolizine and directly elaborated the
molecule into three optically active indolizinylalanine regioisomers. The protocols exploit …

[HTML][HTML] A conserved Neurite Outgrowth and Guidance motif with biomimetic potential in neuronal Cell Adhesion Molecules

G Scapin, M Gasparotto, D Peterle, S Tescari… - Computational and …, 2021‏ - Elsevier
The discovery of conserved protein motifs can, in turn, unveil important regulatory signals,
and when properly designed, synthetic peptides derived from such motifs can be used as …

Development and study of aminocatalyzed asymmetric organic reactions

JM de Carvalho Marques Dourado - 2021‏ - mspace.lib.umanitoba.ca
Chirality is an important feature that many Organic molecules possess and can have huge
repercussions in the activity of Organic compounds. Therefore, the development of …