Substituted 1, 2, 3, 4-tetrahydrocyclopenta [b] indol-3-yl) acetic acid derivatives useful in the treatment of autoimmune and inflammatory disorders
RM Jones, DJ Buzard, S Han, SH Kim… - US Patent …, 2013 - Google Patents
US8580841B2 - Substituted 1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid derivatives
useful in the treatment of autoimmune and inflammatory disorders - Google Patents …
useful in the treatment of autoimmune and inflammatory disorders - Google Patents …
New piperidinylamino-thieno [2, 3-D] pyrimidine compounds
D Dhanoa, O Becker, S Noiman, S Reddy… - US Patent App. 10 …, 2005 - Google Patents
The present invention relates to the discovery of new compounds which are 5-HT
modulators, eg, antago nists, and/or SSRIs, that can be used for treating, preventing or …
modulators, eg, antago nists, and/or SSRIs, that can be used for treating, preventing or …
Processes for the preparation of (R)-2-(7-(4-cyclopentyl-3-(trifluoromethyl) benzyloxy)-1, 2, 3, 4-tetrahydrocyclopenta [b] indol-3-yl) acetic acid and salts thereof
AG Montalban, DJ Buzard, JA DeMattei… - US Patent …, 2014 - Google Patents
PCT Pub. No.: WO2011/094008(57) The present invention relates to processes and
intermediates PCT Pub. Date: Aug. 4, 2011 useful in the preparation of (R)-2-(7-(4 …
intermediates PCT Pub. Date: Aug. 4, 2011 useful in the preparation of (R)-2-(7-(4 …
Substituted tricyclic acid derivatives as S1P1 receptor agonists useful in the treatment of autoimmune and inflammatory disorders
RM Jones, DJ Buzard, AM Kawasaki, SH Kim… - US Patent …, 2013 - Google Patents
The present invention relates to certain substituted tricyclic acid derivatives of Formula (I)
and pharmaceutically accept able salts thereof, which exhibit useful pharmacological …
and pharmaceutically accept able salts thereof, which exhibit useful pharmacological …
Piperidinylamino-thieno [2, 3-D] pyrimidine compounds
DS Dhanoa, O Becker, S Noiman, AS Reddy… - US Patent …, 2009 - Google Patents
The invention relates to 5-HT receptor modulators, particu larly 5-HT, antagonists. Novel
piperidinylamino-thieno2. 3-dipyrimidine compounds represented by Formula I, II and III …
piperidinylamino-thieno2. 3-dipyrimidine compounds represented by Formula I, II and III …
Methods of treating conditions related to the S1P1 receptor
A Glicklich, MMS Kam, WR Shanahan - US Patent 11,007,175, 2021 - Google Patents
Provided are methods of treatment of a sphingosine 1-phos phate subtype 1 (S1P1) receptor-
associated disorder com prising prescribing and/or administering to an individual in need …
associated disorder com prising prescribing and/or administering to an individual in need …
Substituted arylamine compounds and methods of treatment
O Becker, R Melendez, Y Marantz… - US Patent …, 2011 - Google Patents
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Substituted tricyclic acid derivatives as S1P1 receptor agonists useful in the treatment of autoimmune and inflammatory disorders
RM Jones, DJ Buzard, AM Kawasaki, SH Kim… - US Patent …, 2015 - Google Patents
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Continuation of application No. 13/060,477, filed as application No. PCT/US2009/004851 on …
Continuation of application No. 13/060,477, filed as application No. PCT/US2009/004851 on …
S1P receptor modulating compounds and use thereof
2007-07-27 Assigned to AMGEN INC. reassignment AMGEN INC. ASSIGNMENT OF
ASSIGNORS INTEREST (SEE DOCUMENT FOR DETAILS). Assignors: BURLI, ROLAND …
ASSIGNORS INTEREST (SEE DOCUMENT FOR DETAILS). Assignors: BURLI, ROLAND …