Current pharmacotherapy and multi-target approaches for Alzheimer's disease

SL Cheong, JK Tiew, YH Fong, HW Leong, YM Chan… - Pharmaceuticals, 2022 - mdpi.com
Alzheimer's disease (AD) is a neurodegenerative disorder characterized by decreased
synaptic transmission and cerebral atrophy with appearance of amyloid plaques and …

A comprehensive review of multi-target directed ligands in the treatment of Alzheimer's disease

C Pathak, UD Kabra - Bioorganic Chemistry, 2024 - Elsevier
Alzheimer's disease (AD) is the most common form of dementia affecting specifically older
population. AD is an irreversible neurodegenerative CNS disorder associated with complex …

Mannich reaction mediated derivatization of chromones and their biological evaluations as putative multipotent ligands for the treatment of Alzheimer's disease

N Kumar, K Jangid, V Kumar, B Devi, T Arora… - RSC Medicinal …, 2024 - pubs.rsc.org
Alzheimer's disease (AD) is a complex neurological disorder and multiple pathways are
associated with its pathology. Currently available single-targeting drugs are found to be …

Phenylstyrylpyrimidine derivatives as potential multipotent therapeutics for Alzheimer's disease

B Devi, K Jangid, V Kumar, T Arora, N Kumar… - RSC Medicinal …, 2024 - pubs.rsc.org
Alzheimer's disease (AD) is a multifactorial neurological disorder that affects millions of
people worldwide. Despite extensive research efforts, there are currently no effective …

Artificial intelligence assisted identification of potential tau aggregation inhibitors: ligand-and structure-based virtual screening, in silico ADME, and molecular …

B Das, AT Mathew, ATK Baidya, B Devi, RR Salmon… - Molecular Diversity, 2024 - Springer
Alzheimer's disease (AD) is a severe, growing, multifactorial disorder affecting millions of
people worldwide characterized by cognitive decline and neurodegeneration. The …

Design, synthesis, and biological evaluation of novel chromanone derivatives as multifunctional agents for the treatment of Alzheimer's Disease

X Li, T Li, F Zhan, F Cheng, L Lu, B Zhang… - ACS Chemical …, 2022 - ACS Publications
Based on a multitarget strategy, a series of novel chromanone–1-benzyl-1, 2, 3, 6-
tetrahydropyridin hybrids were identified for the potential treatment of Alzheimer's disease …

Design, synthesis and biological evaluation of oxadiazole clubbed piperazine derivatives as potential antidepressant agents

B Sahu, R Bhatia, D Kaur, D Choudhary, R Rawat… - Bioorganic …, 2023 - Elsevier
Piperazine derivatives have been of great interest to medicinal chemists in the development
of antidepressant drugs due to their distinct molecular and structural features along with their …

Calcium channel blockers' contribution to overcoming Current drug discovery challenges in Alzheimer's disease

PJ Bernard, D Bellili, L Ismaili - Expert Opinion on Drug Discovery, 2024 - Taylor & Francis
Introduction Alzheimer's disease (AD) is a progressive, irreversible, and multifactorial brain
disorder that gradually and insidiously destroys individual's memory, thinking, and other …

Design, Synthesis, and Biological Investigation of Quinazoline Derivatives as Multitargeting Therapeutics in Alzheimer's Disease Therapy

A Verma, DK Waiker, N Singh, A Roy… - ACS Chemical …, 2024 - ACS Publications
An efficient and promising method of treating complex neurodegenerative diseases like
Alzheimer's disease (AD) is the multitarget-directed approach. Here in this work, a series of …

Virtual screening and molecular dynamics simulation approach for the identification of potential multi-target directed ligands for the treatment of Alzheimer's disease

K Jangid, B Devi, A Sahoo, V Kumar… - Journal of …, 2024 - Taylor & Francis
Alzheimer's disease (AD) is a multifactorial neurological disorder characterized by memory
loss and cognitive impairment. The currently available single-targeting drugs have miserably …