Histone acetyltransferases CBP/p300 in tumorigenesis and CBP/p300 inhibitors as promising novel anticancer agents

Q Chen, B Yang, X Liu, XD Zhang, L Zhang… - Theranostics, 2022‏ - pmc.ncbi.nlm.nih.gov
The histone acetyltransferases CBP and p300, often referred to as CBP/p300 due to their
sequence homology and functional overlap and co-operation, are emerging as critical …

Transcriptional co-activators: emerging roles in signaling pathways and potential therapeutic targets for diseases

PD Talukdar, U Chatterji - Signal transduction and targeted therapy, 2023‏ - nature.com
Specific cell states in metazoans are established by the symphony of gene expression
programs that necessitate intricate synergic interactions between transcription factors and …

Histone modifications in transcriptional regulation

SL Berger - Current opinion in genetics & development, 2002‏ - Elsevier
Covalent modifications of the amino termini of the core histones in nucleosomes have
important roles in gene regulation. Research in the past two years reveals these …

[HTML][HTML] Acetylation of RelA at discrete sites regulates distinct nuclear functions of NF‐κB

L Chen, Y Mu, WC Greene - The EMBO journal, 2002‏ - embopress.org
The nuclear function of the heterodimeric NF‐κB transcription factor is regulated in part
through reversible acetylation of its RelA subunit. We now demonstrate that the p300 and …

Epigenetics in the pathogenesis of diabetic nephropathy: Epigenetics in the pathogenesis of diabetic nephropathy

X Li, L Lu, W Hou, T Huang, X Chen… - Acta Biochimica et …, 2021‏ - pmc.ncbi.nlm.nih.gov
Diabetic nephropathy (DN), which is a common microvascular complication with a high
incidence in diabetic patients, greatly increases the mortality of patients. With further study …

The SMRT and N-CoR corepressors are activating cofactors for histone deacetylase 3

MG Guenther, ORR Barak, MA Lazar - Molecular and cellular …, 2001‏ - Taylor & Francis
Repression of gene transcription is linked to regulation of chromatin structure through
deacetylation of core histone amino-terminal tails. This action is mediated by histone …

Transcription factor dimerization activates the p300 acetyltransferase

E Ortega, S Rengachari, Z Ibrahim, N Hoghoughi… - Nature, 2018‏ - nature.com
The transcriptional co-activator p300 is a histone acetyltransferase (HAT) that is typically
recruited to transcriptional enhancers and regulates gene expression by acetylating …

CBP and p300: HATs for different occasions

E Kalkhoven - Biochemical pharmacology, 2004‏ - Elsevier
The transcriptional coactivators CREB binding protein (CBP) and p300 are key regulators of
RNA polymerase II-mediated transcription. Genetic alterations in the genes encoding these …

Transcription factors in liver development, differentiation, and regeneration

RH Costa, VV Kalinichenko, AXL Holterman… - Hepatology, 2003‏ - journals.lww.com
Transcriptional Activation. The liver performs essential functions in the body by uniquely
expressing hepatocyte-specific genes encoding plasma proteins, clotting factors and …

Regulating histone acetyltransferases and deacetylases

G Legube, D Trouche - EMBO reports, 2003‏ - embopress.org
Histone acetyltransferases and histone deacetylases regulate the acetylation of histones
and transcription factors, and in doing so have major roles in the control of cell fate. Many …