Adsorption of alprazolam drug on the B12N12 and Al12N12 nano-cages for biological applications: A DFT study

S Kaviani, S Shahab, M Sheikhi - Physica E: Low-dimensional Systems …, 2021‏ - Elsevier
In this study, density functional theory (DFT) calculations were used to investigate the
interaction of the B 12 N 12 and Al 12 N 12 nano-cages with alprazolam (ALP) in the gas …

[HTML][HTML] Novel pyrazolo [3, 4-d] pyrimidines as potential anticancer agents: Synthesis, VEGFR-2 inhibition, and mechanisms of action

Z Ruzi, K Bozorov, L Nie, J Zhao, HA Aisa - Biomedicine & …, 2022‏ - Elsevier
Highlights•Novel tricyclic pyrazolo [3, 4-d] pyrimidine derivatives were synthesized.•
Compound 10k exhibited anticancer activity in vivo.•Compound 10k demonstrated VEGFR-2 …

Discovery of novel coumarin-schiff base hybrids as potential acetylcholinesterase inhibitors: design, synthesis, enzyme inhibition, and computational studies

AH Hasan, FA Abdulrahman, AJ Obaidullah… - Pharmaceuticals, 2023‏ - mdpi.com
To discover anti-acetylcholinesterase agents for the treatment of Alzheimer's disease (AD), a
series of novel Schiff base-coumarin hybrids was rationally designed, synthesized …

Theoretical calculations of molecular descriptors for anticancer activities of 1, 2, 3-triazole-pyrimidine derivatives against gastric cancer cell line (MGC-803): DFT …

RO Oyewole, AK Oyebamiji, B Semire - Heliyon, 2020‏ - cell.com
Abstracts This work used quantum chemical method via DFT to calculate molecular
descriptors for the development of QSAR model to predict bioactivity (IC 50-50% inhibition …

A novel class of phenylpyrazolone-sulphonamides rigid synthetic anticancer molecules selectively inhibit the isoform IX of carbonic anhydrases guided by molecular …

MT Khayat, HEA Ahmed, AM Omar… - Journal of …, 2023‏ - Taylor & Francis
All the previously reported phenylpyrazoles as carbonic anhydrase inhibitors (CAIs) were
found to have small sizes and high levels of flexibility, and hence showed low selectivity …

Screening of natural compounds from Cyperus rotundus Linn against SARS-CoV-2 main protease (Mpro): An integrated computational approach

SB Kumar, S Krishna, S Pradeep, DE Mathews… - Computers in biology …, 2021‏ - Elsevier
Abstract Coronavirus disease 2019 (COVID-19) is a viral respiratory disease that has been
spreading across the globe. The World Health Organization (WHO) declared it as a public …

[HTML][HTML] In-silico exploration and structure-based design of praziquantel derivatives as potential inhibitors of schistosoma mansoni Glutathione S-transferase (SmGST)

SC Jáafaru, A Uzairu, MS Sallau, GI Ndukwe… - Scientific African, 2024‏ - Elsevier
Schistosomiasis is a chronic parasitic disease with significant public health challenges due
to the limited number of treatment options and increasing levels of drug resistance against …

Benzyloxychalcone Hybrids as Prospective Acetylcholinesterase Inhibitors against Alzheimer's Disease: Rational Design, Synthesis, In Silico ADMET Prediction …

HM Al-Maqtari, AH Hasan, M Suleiman… - ACS …, 2024‏ - ACS Publications
Acetylcholinesterase inhibitors (AChEIs) are crucial therapeutic targets for both the early and
severe stages of Alzheimer's disease (AD). Chalcones and their chromone-based …

Assessment of the adsorption mechanism of amantadine drug onto pristine, Si-and Ge-doped Al12N12, and Al12P12 nanocages: A comparative DFT study

M Kamel, EAM Saleh, K Mohammadifard… - Materials Chemistry and …, 2023‏ - Elsevier
In the current study, the adsorption characteristics of pristine and doped (Si and Ge)-Al 12 N
12 (AlN) and Al 12 P 12 (AlP) nanocages towards the amantadine (AM) drug have been …

DFT and molecular simulation validation of the binding activity of PDEδ inhibitors for repression of oncogenic k-Ras

TA Majrashi, A Sabt, H Almahli, MA El Hassab… - PLoS …, 2024‏ - journals.plos.org
The development of effective drugs targeting the K-Ras oncogene product is a significant
focus in anticancer drug development. Despite the lack of successful Ras signaling …