Discovery of 2-(4-(2-fluoroethoxy) piperidin-1-yl)-9-methyl-9H-pyrrolo [2, 3-b: 4, 5-c'] dipyridine ([18F] PI-2014) as PET tracer for the detection of pathological …

E Gabellieri, F Capotosti, J Molette… - European journal of …, 2020 - Elsevier
The compound screening was initiated with a direct staining assay to identify compounds
binding to Tau aggregates and not Abeta plaques using human brain sections derived from …

Exploring the Propensities of Fluorescent Carbazole Analogs toward the Inhibition of Amyloid Aggregation in Type 2 Diabetes: An Experimental and Theoretical …

T Mallick, A Karmakar, A Mukhuty… - The Journal of …, 2021 - ACS Publications
Amyloid aggregation is a pathological trait observed in many incurable and fatal
neurodegenerative and metabolic diseases associated with misfolding and self-assembly of …

9H-pyrrolo-dipyridine derivatives

J Mercier, L Provins, C Vermeiren… - US Patent 11,312,716, 2022 - Google Patents
US11312716B2 - 9H-pyrrolo-dipyridine derivatives - Google Patents US11312716B2 - 9H-pyrrolo-dipyridine
derivatives - Google Patents 9H-pyrrolo-dipyridine derivatives Download PDF Info …

Azaindole compounds as histone methyltransferase inhibitors

C Yu, M Yu, M Zancanella, Z Li - US Patent 11,111,243, 2021 - Google Patents
The present disclosure provides certain angular tricyclic compounds that are histone
methyltransferases G9a and/or GLP inhibitors and are therefore useful for the treatment of …

Histone methyltransferase inhibitors

M Yu, Z Li - US Patent 11,713,299, 2023 - Google Patents
Wang et al.,“Histone H3K9 methyltransferase G9a represses PPARy expression and
adipogenesis” EMBO J.(2013) 32 (1) 45-59. Yang et al.,“G9a coordinates with the RPA …

Histone methyltransferase inhibitors

M Yu, Z Li - US Patent 10,829,452, 2020 - Google Patents
DSUUMHAYXBBFLM-UHFFFAOYSA-N COC1= C (OCCCN2CCCC2) C= C2N= C (NC
(C)(C) C) C3= C (CCC3) C2= C1 Chemical compound COC1= C (OCCCN2CCCC2) C …