Heterocyclic scaffolds: centrality in anticancer drug development
Cancer has been cursed for human beings for long time. Millions people lost their lives due
to cancer. Despite of the several anticancer drugs available, cancer cannot be cured; …
to cancer. Despite of the several anticancer drugs available, cancer cannot be cured; …
Application of Palladium Based Precatalytic Systems in the Suzuki‐Miyaura Cross‐Coupling Reactions of Chloro‐Heterocycles
Carbon‐Carbon bond forming reactions using Suzuki‐Miyaura cross‐coupling (SMC)
technology to construct aryl‐aryl, aryl‐heteroaryl or heteroaryl‐heteroaryl linkages continues …
technology to construct aryl‐aryl, aryl‐heteroaryl or heteroaryl‐heteroaryl linkages continues …
Visible-light-induced, metal-free carbene insertion into B–H bonds between acylsilanes and pinacolborane
JH Ye, L Quach, T Paulisch… - Journal of the American …, 2019 - ACS Publications
Carbene insertion reactions with B–H bonds are a challenging but promising method for the
synthesis of organoboranes. Herein, we report visible-light-induced B–H insertions of HBpin …
synthesis of organoboranes. Herein, we report visible-light-induced B–H insertions of HBpin …
Suzuki-Miyaura cross-coupling of unprotected, nitrogen-rich heterocycles: Substrate scope and mechanistic investigation
MA Düfert, KL Billingsley… - Journal of the American …, 2013 - ACS Publications
The Suzuki-Miyaura cross-coupling of unprotected, nitrogen-rich heterocycles using
precatalysts P1 or P2 is reported. The procedure allows for the reaction of variously …
precatalysts P1 or P2 is reported. The procedure allows for the reaction of variously …
Nickel-catalyzed Suzuki–Miyaura coupling of aliphatic amides
We report the Ni-catalyzed Suzuki–Miyaura coupling of aliphatic amide derivatives. Prior
studies have shown that aliphatic amide derivatives can undergo Ni-catalyzed carbon …
studies have shown that aliphatic amide derivatives can undergo Ni-catalyzed carbon …
Biosynthesis, characterization and catalytic activity of an Ag/zeolite nanocomposite for base-and ligand-free oxidative hydroxylation of phenylboronic acid and …
This paper reports on the synthesis and use of an Ag/zeolite nanocomposite as a separable
catalyst for the ligand-free hydroxylation of phenylboronic acid to phenol and the reduction …
catalyst for the ligand-free hydroxylation of phenylboronic acid to phenol and the reduction …
Micellar system in copper-catalysed hydroxylation of arylboronic acids: facile access to phenols
K Inamoto, K Nozawa, M Yonemoto… - Chemical …, 2011 - pubs.rsc.org
Micellar system in copper-catalysed hydroxylation of arylboronic acids: facile access to phenols -
Chemical Communications (RSC Publishing) DOI:10.1039/C1CC14974A Royal Society of …
Chemical Communications (RSC Publishing) DOI:10.1039/C1CC14974A Royal Society of …
Palladium-catalyzed C–O bond formation: direct synthesis of phenols and aryl/alkyl ethers from activated aryl halides
G Chen, ASC Chan, FY Kwong - Tetrahedron Letters, 2007 - Elsevier
A simple and efficient palladium-catalyzed carbon–oxygen bond formation is reported. The
palladium-tri-tert-butylphosphine complex was found to be effective in converting …
palladium-tri-tert-butylphosphine complex was found to be effective in converting …
Nitrogen-carbon bond formation from N2 and CO2 promoted by a hafnocene dinitrogen complex yields a substituted hydrazine
WH Bernskoetter, E Lobkovsky… - Angewandte Chemie …, 2007 - collaborate.princeton.edu
Abstract (Chemical Equation Presented) Hafnocene and hydrazine: The addition of two
equivalents of carbon dioxide to the hafnocene dinitrogen complex 1 proved effective for the …
equivalents of carbon dioxide to the hafnocene dinitrogen complex 1 proved effective for the …
Mechanistic Studies and Data Science-Guided Exploration of Bromotetrazine Cross-Coupling
A thorough mechanistic investigation of the Pd-catalyzed and Ag-mediated cross-coupling of
the monosubstituted tetrazine 3-bromo-1, 2, 4, 5-tetrazine with boronic acids is reported. The …
the monosubstituted tetrazine 3-bromo-1, 2, 4, 5-tetrazine with boronic acids is reported. The …