Luteolin, a flavone ingredient: Anticancer mechanisms, combined medication strategy, pharmacokinetics, clinical trials, and pharmaceutical researches

M Shi, Z Chen, H Gong, Z Peng, Q Sun… - Phytotherapy …, 2024‏ - Wiley Online Library
Current pharmaceutical research is energetically excavating the pharmacotherapeutic role
of herb‐derived ingredients in multiple malignancies' targeting. Luteolin is one of the major …

Heme-thiolate monooxygenase cytochrome P450 1B1, an old dog with many new tricks

JW Kim, HC Tung, B Yang, R Pant, X Guan… - Pharmacological …, 2025‏ - Elsevier
ABSTRACT Cytochrome P450 (CYP) 1B1 is a heme-thiolate monooxygenase traditionally
recognized for its xenobiotic functions and extrahepatic expressions. Recent studies have …

Urolithin A increases the natural killer activity of PBMCs in patients with prostate cancer

V Rogovskii, VV Murugin, N Vorobyev… - Frontiers in …, 2025‏ - frontiersin.org
Background The natural killer (NK) activity of peripheral blood mononuclear cells (PBMCs)
is a crucial defense against the onset and spread of cancer. Studies have shown that …

[HTML][HTML] In Silico Exploration of AHR-HIF Pathway Interplay: Implications for Therapeutic Targeting in ccRCC

F Gregoris, G Minervini, SCE Tosatto - Genes, 2024‏ - mdpi.com
The oxygen-sensing pathway is a crucial regulatory circuit that defines cellular conditions
and is extensively exploited in cancer development. Pathogenic mutations in the von Hippel …

Clofazimine inhibits small-cell lung cancer progression by modulating the kynurenine/aryl hydrocarbon receptor axis

G Sharma, KM Abdullah, FA Qais, P Khan… - International Journal of …, 2024‏ - Elsevier
Small cell lung cancer (SCLC) is one of the highly metastatic malignancies that contributes
to∼ 15% of all lung cancers. Most SCLC patients (50–60%) develop osteolytic bone …

A pyrazolopyridine as a novel AhR signaling activator with anti-breast cancer properties in vitro and in vivo

MS Abduh, OI Alwassil, SM Aldaqal… - Biochemical …, 2024‏ - Elsevier
Breast cancer is one of the main causes of malignancy-related deaths globally and has a
significant impact on women's quality of life. Despite significant therapeutic advances, there …

[HTML][HTML] Discovery of a novel AhR–CYP1A1 axis activator for mitigating inflammatory diseases using an in situ functional imaging assay

F Zhang, B Zhao, Y Fan, L Qin, J Shi, L Chen… - … Pharmaceutica Sinica B, 2025‏ - Elsevier
The aryl hydrocarbon receptor (AhR) plays a crucial role in regulating many physiological
processes. Activating the AhR–CYP1A1 axis has emerged as a novel therapeutic strategy …

Unveiling the Immune effects of AHR in tumors: a decade of insights from bibliometric analysis (2010–2023)

A **e, T Wang, W Shi, F He, X Sun, P Li - Discover Oncology, 2024‏ - Springer
Abstract Background The Aryl Hydrocarbon Receptor (AHR) is a transcription factor that
regulates several biological processes. Its potential in anti-tumor immunotherapy is …

Carbidopa and ZnCarbidopa Induce Reductive Stress in MDA‐MB‐231 Cells

AB Actis Dato, LG Naso, VR Martínez, EG Ferrer… - ChemPlusChem‏ - Wiley Online Library
The redox imbalance, caused by depletion or generation of reactive oxygen species (ROS),
is a key mechanism by which metal complexes exert anticancer effects. Carbidopa has …