Recent advances bioactive 1, 2, 4-triazole-3-thiones

ŞG Küçükgüzel, P Çıkla-Süzgün - European journal of medicinal chemistry, 2015 - Elsevier
Triazoles are heterocyclic compounds which have a five-membered ring of two carbon
atoms and three nitrogen atoms. These structures have been interest in the development of …

A review on 'triazoles': Their chemistry, synthesis and pharmacological potentials

D Dixit, PK Verma, RK Marwaha - Journal of the Iranian Chemical Society, 2021 - Springer
Heterocyclic compounds are cyclic compounds as an atom of ring members with at least two
different elements. In the five-membered aromatic azole chain, triazole compounds …

Chemistry and biological activities of 1, 2, 4-triazolethiones—antiviral and anti-infective drugs

AA Aly, A A. Hassan, MM Makhlouf, S Bräse - Molecules, 2020 - mdpi.com
Mercapto-substituted 1, 2, 4-triazoles are very interesting compounds as they play an
important role in chemopreventive and chemotherapeutic effects on cancer. In recent …

In vitro cytotoxic and in vivo antitumoral activities of some aminomethyl derivatives of 2, 4‐dihydro‐3H‐1, 2, 4‐triazole‐3‐thiones—Evaluation of their …

İ Timur, ÜM Kocyigit, T Dastan, S Sandal… - … of biochemical and …, 2019 - Wiley Online Library
Abstract The 1, 2, 4‐triazole and its derivatives were reported to exhibit various
pharmacological activities such as antimicrobial, analgesic, anti‐inflammatory, antitumoural …

Molecular science for drug development and biomedicine

WZ Zhong, SF Zhou - International journal of molecular sciences, 2014 - mdpi.com
With the avalanche of biological sequences generated in the postgenomic age, molecular
science is facing an unprecedented challenge, ie, how to timely utilize the huge amount of …

[HTML][HTML] Thiazole, triazole, thio-and semicarbazone derivatives-Promising moieties for drug development for the treatment of tuberculosis

CB Scarim, FR Pavan - European Journal of Medicinal Chemistry Reports, 2021 - Elsevier
Thiazole, triazole, thio and semicarbazones are privileged motifs that act as
pharmacophores in bioactive compounds for various diseases, such as Tuberculosis (TB) …

Synthesis, characterization, linear and NLO properties of novel N-(2, 4-dinitrobenzylidene)-3-chlorobenzenamine schiff base: combined experimental and DFT …

A Benmohammed, D Hadji, A Guendouzi… - Journal of Electronic …, 2021 - Springer
This study entails two parts: The first reports on the synthesis of a novel N-(2, 4-
dinitrobenzylidene)-3-chlorobenzenamine Schiff base and its analysis by ultraviolet–visible …

Tautomerism and structure of azoles: nuclear magnetic resonance spectroscopy

LI Larina - Advances in heterocyclic chemistry, 2018 - Elsevier
This review provides comprehensive data (from the author's work and the literature) on
tautomerism of pyrazoles, imidazoles, 1, 2, 3-and 1, 2, 4-triazoles, tetrazoles …

Facile synthesis, pharmacological and In silico analysis of succinimide derivatives: An approach towards drug discovery

J Rasgania, R Gavadia, K Jakhar - Journal of Molecular Structure, 2023 - Elsevier
The hybrid heterocyclic scaffolds possess extensive medicinal values and significant
pharmaceutical usage. A series of N-substituted-2, 5-dioxopyrrolidine carboxamides …

Synthesis, biological evaluation and molecular dynamics studies of 1, 2, 4-triazole clubbed Mannich bases

VM Patel, NB Patel, MJ Chan-Bacab… - Computational biology and …, 2018 - Elsevier
The present work highlightsthe synthesis of a newer biologically active Mannich bases
contributing 4-((4-fluorobenzylidene) amino)-5-(pyridin-4-yl)-4H-1, 2, 4-triazole-3-thiol and …