Computer-aided multi-objective optimization in small molecule discovery

JC Fromer, CW Coley - Patterns, 2023 - cell.com
Molecular discovery is a multi-objective optimization problem that requires identifying a
molecule or set of molecules that balance multiple, often competing, properties. Multi …

Reinforcement learning for generative ai: A survey

Y Cao, QZ Sheng, J McAuley, L Yao - arxiv preprint arxiv:2308.14328, 2023 - arxiv.org
Deep Generative AI has been a long-standing essential topic in the machine learning
community, which can impact a number of application areas like text generation and …

Coarsenconf: Equivariant coarsening with aggregated attention for molecular conformer generation

D Reidenbach, AS Krishnapriyan - Journal of Chemical …, 2024 - ACS Publications
Molecular conformer generation (MCG) is an important task in cheminformatics and drug
discovery. The ability to efficiently generate low-energy 3D structures can avoid expensive …

Scalable fragment-based 3d molecular design with reinforcement learning

D Flam-Shepherd, A Zhigalin… - arxiv preprint arxiv …, 2022 - arxiv.org
Machine learning has the potential to automate molecular design and drastically accelerate
the discovery of new functional compounds. Towards this goal, generative models and …

Improving small molecule generation using mutual information machine

D Reidenbach, M Livne, RK Ilango, M Gill… - arxiv preprint arxiv …, 2022 - arxiv.org
We address the task of controlled generation of small molecules, which entails finding novel
molecules with desired properties under certain constraints (eg, similarity to a reference …

Target-specific novel molecules with their recipe: Incorporating synthesizability in the design process

SR Krishnan, N Bung, R Srinivasan, A Roy - Journal of Molecular Graphics …, 2024 - Elsevier
Application of Artificial intelligence (AI) in drug discovery has led to several success stories
in recent times. While traditional methods mostly relied upon screening large chemical …

Using Artificial Intelligence for de novo Drug Design and Retrosynthesis

R Arora, N Brosse, C Descamps… - Computational Drug …, 2024 - Wiley Online Library
Artificial intelligence (AI), driven by progress in deep learning, has emerged as a disruptive
technology across multiple industries. The development of AI approaches to de novo drug …

Scalable Fragment-Based 3D Molecular Design with Reinforcement Learning

A Zhigalin - 2023 - dash.harvard.edu
Machine learning has the potential to automate molecular design and drastically accelerate
the discovery of new functional compounds. Towards this goal, generative models and …

Similarity-Driven Regularization for Aligning Chemical and Latent Spaces in Molecular Design

J Yang, T Ma, Y **ao, Y Liu, Y Liu - openreview.net
Generative models play a pivotal role in molecular design by effectively generating target
molecules. Among these, generative models with latent space stand out due to their robust …