[HTML][HTML] Leukemic stem cells and therapy resistance in acute myeloid leukemia

P Stelmach, A Trumpp - Haematologica, 2023 - ncbi.nlm.nih.gov
A major obstacle in the treatment of acute myeloid leukemia (AML) is refractory disease or
relapse after achieving remission. The latter arises from a few therapy-resistant cells within …

Amino acid depletion therapies: starving cancer cells to death

M Butler, LT van der Meer, FN van Leeuwen - Trends in Endocrinology & …, 2021 - cell.com
Targeting tumor cell metabolism is an attractive form of therapy, as it may enhance treatment
response in therapy resistant cancers as well as mitigate treatment-related toxicities by …

Fatty acid metabolism underlies venetoclax resistance in acute myeloid leukemia stem cells

BM Stevens, CL Jones, DA Pollyea, R Culp-Hill… - Nature cancer, 2020 - nature.com
Venetoclax with azacitidine (ven/aza) has emerged as a promising treatment regimen for
acute myeloid leukemia (AML), with a high percentage of clinical remissions in newly …

Venetoclax and azacitidine compared with induction chemotherapy for newly diagnosed patients with acute myeloid leukemia

EM Cherry, D Abbott, M Amaya, C McMahon… - Blood …, 2021 - ashpublications.org
Venetoclax (ven) plus azacitidine (aza) is the standard of care for patients with newly
diagnosed acute myeloid leukemia (AML) who are not candidates for intensive …

Targeting multiple signaling pathways: the new approach to acute myeloid leukemia therapy

JL Carter, K Hege, J Yang, HA Kalpage, Y Su… - Signal transduction and …, 2020 - nature.com
Acute myeloid leukemia (AML) is the most common form of acute leukemia in adults and the
second most common form of acute leukemia in children. Despite this, very little …

Bone marrow mesenchymal stem cells support acute myeloid leukemia bioenergetics and enhance antioxidant defense and escape from chemotherapy

D Forte, M García-Fernández, A Sanchez-Aguilera… - Cell metabolism, 2020 - cell.com
Like normal hematopoietic stem cells, leukemic stem cells depend on their bone marrow
(BM) microenvironment for survival, but the underlying mechanisms remain largely …

APR-246 induces early cell death by ferroptosis in acute myeloid leukemia

R Birsen, C Larrue, J Decroocq, N Johnson… - …, 2021 - pmc.ncbi.nlm.nih.gov
APR-246 is a promising new therapeutic agent that targets p53 mutated proteins in
myelodysplastic syndromes and in acute myeloid leukemia (AML). APR-246 reactivates the …

Metabolic dysregulation contributes to the progression of Alzheimer's disease

X Yan, Y Hu, B Wang, S Wang, X Zhang - Frontiers in neuroscience, 2020 - frontiersin.org
Alzheimer's disease (AD) is an incurable neurodegenerative disease. Numerous studies
have demonstrated a critical role for dysregulated glucose metabolism in its pathogenesis …

Eprenetapopt triggers ferroptosis, inhibits NFS1 cysteine desulfurase, and synergizes with serine and glycine dietary restriction

KM Fujihara, BZ Zhang, TD Jackson, MO Ogunkola… - Science …, 2022 - science.org
The mechanism of action of eprenetapopt (APR-246, PRIMA-1MET) as an anticancer agent
remains unresolved, although the clinical development of eprenetapopt focuses on its …

Mitochondrial inhibitors circumvent adaptive resistance to venetoclax and cytarabine combination therapy in acute myeloid leukemia

C Bosc, E Saland, A Bousard, N Gadaud, M Sabatier… - Nature cancer, 2021 - nature.com
Therapy resistance represents a major clinical challenge in acute myeloid leukemia (AML).
Here we define a 'MitoScore'signature, which identifies high mitochondrial oxidative …