Towards reproducible computational drug discovery

N Schaduangrat, S Lampa, S Simeon… - Journal of …, 2020 - Springer
The reproducibility of experiments has been a long standing impediment for further scientific
progress. Computational methods have been instrumental in drug discovery efforts owing to …

Memory-assisted reinforcement learning for diverse molecular de novo design

T Blaschke, O Engkvist, J Bajorath, H Chen - Journal of cheminformatics, 2020 - Springer
In de novo molecular design, recurrent neural networks (RNN) have been shown to be
effective methods for sampling and generating novel chemical structures. Using a technique …

Human-in-the-loop assisted de novo molecular design

I Sundin, A Voronov, H **ao, K Papadopoulos… - Journal of …, 2022 - Springer
A de novo molecular design workflow can be used together with technologies such as
reinforcement learning to navigate the chemical space. A bottleneck in the workflow that …

Industry-scale application and evaluation of deep learning for drug target prediction

N Sturm, A Mayr, T Le Van, V Chupakhin… - Journal of …, 2020 - Springer
Artificial intelligence (AI) is undergoing a revolution thanks to the breakthroughs of machine
learning algorithms in computer vision, speech recognition, natural language processing …

Human-in-the-loop active learning for goal-oriented molecule generation

Y Nahal, J Menke, J Martinelli, M Heinonen… - Journal of …, 2024 - Springer
Machine learning (ML) systems have enabled the modelling of quantitative structure–
property relationships (QSPR) and structure-activity relationships (QSAR) using existing …

Enhancing reaction-based de novo design using a multi-label reaction class recommender

GM Ghiandoni, MJ Bodkin, B Chen, D Hristozov… - Journal of Computer …, 2020 - Springer
Reaction-based de novo design refers to the in-silico generation of novel chemical
structures by combining reagents using structural transformations derived from known …

TNFipred: a classification model to predict TNF-α inhibitors

NK Prabha, A Sharma, H Sandhu, P Garg - Molecular Diversity, 2024 - Springer
Rheumatoid arthritis (RA), characterized by severe inflammation in the joint lining, is a
progressive, chronic, autoimmune disorder with high morbidity and mortality rates. There are …

Direct steering of de novo molecular generation using descriptor conditional recurrent neural networks (crnns)

PC Kotsias, J Arús-Pous, H Chen, O Engkvist… - 2019 - chemrxiv.org
Deep learning has acquired considerable momentum over the past couple of years in the
domain of de-novo drug design. Particularly, transfer and reinforcement learning have …