Machine learning directed drug formulation development

P Bannigan, M Aldeghi, Z Bao, F Häse… - Advanced Drug Delivery …, 2021‏ - Elsevier
Abstract Machine learning (ML) has enabled ground-breaking advances in the healthcare
and pharmaceutical sectors, from improvements in cancer diagnosis, to the identification of …

Merging ligand-based and structure-based methods in drug discovery: an overview of combined virtual screening approaches

J Vázquez, M López, E Gibert, E Herrero, FJ Luque - Molecules, 2020‏ - mdpi.com
Virtual screening (VS) is an outstanding cornerstone in the drug discovery pipeline. A variety
of computational approaches, which are generally classified as ligand-based (LB) and …

A de novo molecular generation method using latent vector based generative adversarial network

O Prykhodko, SV Johansson, PC Kotsias… - Journal of …, 2019‏ - Springer
Deep learning methods applied to drug discovery have been used to generate novel
structures. In this study, we propose a new deep learning architecture, LatentGAN, which …

SMILES-based deep generative scaffold decorator for de-novo drug design

J Arús-Pous, A Patronov, EJ Bjerrum, C Tyrchan… - Journal of …, 2020‏ - Springer
Molecular generative models trained with small sets of molecules represented as SMILES
strings can generate large regions of the chemical space. Unfortunately, due to the …

Improving Chemical Autoencoder Latent Space and Molecular De Novo Generation Diversity with Heteroencoders

EJ Bjerrum, B Sattarov - Biomolecules, 2018‏ - mdpi.com
Chemical autoencoders are attractive models as they combine chemical space navigation
with possibilities for de novo molecule generation in areas of interest. This enables them to …

Virtual screening web servers: designing chemical probes and drug candidates in the cyberspace

N Singh, L Chaput, BO Villoutreix - Briefings in bioinformatics, 2021‏ - academic.oup.com
The interplay between life sciences and advancing technology drives a continuous cycle of
chemical data growth; these data are most often stored in open or partially open databases …

Practical guidelines for the use of gradient boosting for molecular property prediction

D Boldini, F Grisoni, D Kuhn, L Friedrich… - Journal of …, 2023‏ - Springer
Decision tree ensembles are among the most robust, high-performing and computationally
efficient machine learning approaches for quantitative structure–activity relationship (QSAR) …

Advances with support vector machines for novel drug discovery

VG Maltarollo, T Kronenberger… - Expert opinion on …, 2019‏ - Taylor & Francis
Introduction: Novel drug discovery remains an enormous challenge, with various computer-
aided drug design (CADD) approaches having been widely employed for this purpose …

[HTML][HTML] Alkaloids in contemporary drug discovery to meet global disease needs

S Daley, GA Cordell - Molecules, 2021‏ - mdpi.com
An overview is presented of the well-established role of alkaloids in drug discovery, the
application of more sustainable chemicals, and biological approaches, and the …

Sensing and sensitivity: Computational chemistry of graphene‐based sensors

A Piras, C Ehlert, G Gryn'ova - Wiley Interdisciplinary Reviews …, 2021‏ - Wiley Online Library
Highly efficient, tunable, biocompatible, and environmentally friendly electrochemical
sensors featuring graphene‐based materials pose a formidable challenge for computational …