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An appraisal of anti-mycobacterial activity with structure-activity relationship of piperazine and its analogues: A review
Piperazine, is privileged six membered nitrogen containing heterocyclic ring also known as
1, 4-Diazacyclohexane. Consequently, piperazine is a versatile medicinally important …
1, 4-Diazacyclohexane. Consequently, piperazine is a versatile medicinally important …
Recent advancements and developments in search of anti-tuberculosis agents: a quinquennial update and future directions
Tuberculosis (TB) has been considered as the highly chronic, contagious and infectious
disorder caused by Mycobacterium tuberculosis (Mtb). Every year more than 10 million …
disorder caused by Mycobacterium tuberculosis (Mtb). Every year more than 10 million …
Synthesis, antituberculosis studies and biological evaluation of new quinoline derivatives carrying 1, 2, 4-oxadiazole moiety
TG Shruthi, S Eswaran, P Shivarudraiah… - Bioorganic & medicinal …, 2019 - Elsevier
Tuberculosis is the infectious disease caused by mycobacterium tuberculosis (Mtb),
responsible for the utmost number of deaths annually across the world. Herein, twenty-one …
responsible for the utmost number of deaths annually across the world. Herein, twenty-one …
An insight into the biological activity and structure-based drug design attributes of sulfonylpiperazine derivatives
The development of new, effective drugs containing nitrogen and sulfur heteroatoms is of
paramount importance in medicinal chemistry. A versatile and rational approach for drug …
paramount importance in medicinal chemistry. A versatile and rational approach for drug …
Discovery and characterization of antimycobacterial nitro-containing compounds with distinct mechanisms of action and in vivo efficacy
Nitro-containing compounds have emerged as important agents in the control of
tuberculosis (TB). From a whole-cell high-throughput screen for Mycobacterium tuberculosis …
tuberculosis (TB). From a whole-cell high-throughput screen for Mycobacterium tuberculosis …
New structural classes of antituberculosis agents
Tuberculosis (TB), one of the deadliest diseases is shattering the health and socioeconomic
status of the society. The emergence of multidrug resistant (MDR) and extremely drug …
status of the society. The emergence of multidrug resistant (MDR) and extremely drug …
Current development of 5-nitrofuran-2-yl derivatives as antitubercular agents
Pulmonary tuberculosis (TB) is an infectious disease caused by Mycobacterium tuberculosis
(MTB) and still remains one of the foremost fatal infectious diseases, infecting nearly a third …
(MTB) and still remains one of the foremost fatal infectious diseases, infecting nearly a third …
Identification of nitrofuranylchalcone tethered benzoxazole-2-amines as potent inhibitors of drug resistant Mycobacterium tuberculosis demonstrating bactericidal …
Ever increasing drug resistance has become an impeding threat that continues to hamper
effective tackling of otherwise treatable tuberculosis (TB). Such dismal situation necessitates …
effective tackling of otherwise treatable tuberculosis (TB). Such dismal situation necessitates …
The optimization and characterization of functionalized sulfonamides derived from sulfaphenazole against Mycobacterium tuberculosis with reduced CYP 2C9 …
H Chen, B Wang, P Li, H Yan, G Li, H Huang… - Bioorganic & Medicinal …, 2021 - Elsevier
In this study, a series of sulfonamide compounds was designed and synthesized through the
systematic optimization of the antibacterial agent sulfaphenazole for the treatment of …
systematic optimization of the antibacterial agent sulfaphenazole for the treatment of …
Synthesis, evaluation and CoMFA/CoMSIA study of nitrofuranyl methyl N-heterocycles as novel antitubercular agents
A Wang, Y Yang, Y Jun, B Wang, K Lv, M Liu… - Bioorganic & medicinal …, 2018 - Elsevier
A series of novel nitrofuranyl methyl N-heterocycles based on the structure of IIIM-MCD-211
were designed and synthesized. Compounds 6d, 8b and 12a show excellent activity against …
were designed and synthesized. Compounds 6d, 8b and 12a show excellent activity against …