Design, classification, and adverse effects of NSAIDs: A review on recent advancements

M Arfeen, A Srivastava, N Srivastava, RA Khan… - Bioorganic & Medicinal …, 2024‏ - Elsevier
Inflammation is a hallmark of many diseases, including cancer, neurodegenerative diseases
like Alzheimer's, type II diabetes, rheumatoid arthritis, and asthma. Nonsteroidal anti …

Selective COX-2 inhibitors as anticancer agents: a patent review (2018-2023)

M Mahboubi-Rabbani, AH Abdolghaffari… - Expert Opinion on …, 2024‏ - Taylor & Francis
Introduction COX-2 is a crucial enzyme in the manufacture of prostaglandins. The enzyme's
metabolites might have an important function as regulators of the inflammatory response …

Optimizing bioreactor conditions for Spirulina fermentation by Lactobacillus helveticus and Kluyveromyces marxianus: Impact on chemical & bioactive properties

C Yay, ZO Cinar, S Donmez, TB Tumer, O Guneser… - Bioresource …, 2024‏ - Elsevier
This study focused on optimizing the production of fermented Spirulina (FS) products using a
bioactivity-guided strategy with Lactobacillus helveticus B-4526 and Kluyveromyces …

Novel tryptanthrin derivatives with benzenesulfonamide substituents: Design, synthesis, and anti-inflammatory evaluation

J Du, P Liu, Y Zhu, G Wang, S **ng, T Liu, J **a… - European Journal of …, 2023‏ - Elsevier
Herein, two series of tryptanthrin derivatives with benzenesulfonamide substituents were
designed and synthesized to discover novel anti-inflammatory agents. The anti-inflammatory …

Novel thiadiazol derivatives; design, synthesis, biological activity, molecular docking and molecular dynamics

D Osmaniye, AE Evren, Ş Karaca, Y Özkay… - Journal of Molecular …, 2023‏ - Elsevier
Currently, selective COX-2 inhibitors are used as a novel alternative approach in the course
of pain management due to their reduced adverse that generally occur after COX-1 …

Discovery of novel deoxyvasicinone derivatives with benzenesulfonamide substituents as multifunctional agents against Alzheimer's disease

S Dong, J **a, F Wang, L Yang, S **ng, J Du… - European Journal of …, 2024‏ - Elsevier
A series of deoxyvasicinone derivatives with benzenesulfonamide substituents were
designed and synthesized to find a multifunctional anti-Alzheimer's disease (AD) drug. The …

Novel analytical sensing strategy using a palladium nanomaterial-based electrode for nimesulide electrochemical reduction

RB Goularte, JP Winiarski, E Latocheski… - Journal of …, 2022‏ - Elsevier
Nimesulide (NIM) is a non-steroidal anti-inflammatory drug considered an emerging
contaminant. Thus, a novel sensing platform composed of an ionic silsesquioxane material …

Novel quinoline-based derivatives: A new class of PDE4B inhibitors for adjuvant-induced arthritis

S **ng, W Fan, J Chen, J Du, T Liu, S Dong… - European Journal of …, 2022‏ - Elsevier
A total of 31 quinoline-based derivatives were designed and synthesized to develop novel
anti-inflammatory drugs. After the toxicity of synthetic compounds to RAW264. 7 cells were …

Novel nimesulide multicomponent solid forms: screening, synthesis, thermoanalytical study and characterization

AC de Almeida, PO Ferreira, MV Porto… - Journal of Thermal …, 2024‏ - Springer
Nimesulide (NMS) is a widely used non-steroidal anti-inflammatory drug, however, presents
low aqueous solubility. One way to overcome the solubility issue of drugs is altering their …

Synergy between cyclooxygenase-2 inhibitors and hyaluronic acid in the treatment of osteoarthritis: Illumination of signaling cascade, nanotechnology-driven delivery …

S Thote, P Gorella, S Arya, A Mourya… - Journal of Drug Delivery …, 2024‏ - Elsevier
Osteoarthritis (OA) is generally caused by a variety of risk factors, the most notable of which
are growing age and obesity. Pathophysiologically, chondrocytes alter their morphology and …