Recent advances in the synthesis of pyrido [1, 2-a] indoles

Y Yao, M Alami, A Hamze, O Provot - Organic & Biomolecular …, 2021 - pubs.rsc.org
The pyrido [1, 2-a] indole unit found in many organic compounds such as natural products,
pharmaceuticals, and materials, has intensively stimulated the research of new synthetic …

Rational synthetic methods in creating promising (hetero) aromatic molecules and materials

GV Zyryanov, DS Kopchuk, IS Kovalev, S Santra… - Mendeleev …, 2020 - Elsevier
In this focus article, the recent syntheses of various (hetero) aromatic/macrocyclic
molecules/scaffolds such as (thia) calixarenes, iptycenes,[poly](aza) arenes, 2, 2 …

Silver-catalyzed [3+ 3] dipolar cycloaddition of trifluorodiazoethane and glycine imines: access to highly functionalized trifluoromethyl-substituted triazines and …

Z Chen, N Ren, X Ma, J Nie, FG Zhang, JA Ma - ACS Catalysis, 2019 - ACS Publications
Herein we disclose a silver-catalyzed [3+ 3] 1, 3-dipolar cycloaddition reaction of
trifluorodiazoethane with glycine imines. This reaction exhibits manifold remarkable …

Copper-Catalyzed Cascade Cyclization Reaction of Enamines and Electron-Deficient Terminal Alkynes: Synthesis of Polysubstituted Pyrido[1,2-a]indoles

P Liu, M Yang, Y Gong, Y Yu, YL Zhao - Organic letters, 2019 - ACS Publications
A novel copper-catalyzed cascade cyclization reaction between enamines and electron-
deficient terminal alkynes has been developed. The reaction provides a new and efficient …

Nucleophilic substitution of hydrogen–the Boger reaction sequence as an approach towards 8-(pyridin-2-yl) coumarins

RF Fatykhov, MI Savchuk, ES Starnovskaya… - Mendeleev …, 2019 - mathnet.ru
5, 7-Dimethoxy-8-(3, 6-diphenylpyridin-2-yl) coumarins were obtained from 5, 7-
dimethoxycoumarins and 3, 6-diphenyl-1, 2, 4-triazines via the protocol comprising aromatic …

Synthesis of Benzo[b]fluoranthenes and Spiroacridines from Fluorene-Derived Alkenes and N-Arylimines via a Tandem Reaction with Benzynes

W Wang, H Wan, G Du, B Dai, L He - Organic letters, 2019 - ACS Publications
Two tandem processes involving the cycloaddition of benzynes have been developed for
the synthesis of polyaromatic hydrocarbons. Benzynes react with fluorene-derived alkenes …

Synthesis of 5-Phenyl-2, 2'-bipyridines 6-Substituted with Donor Groups by aza-Diels–Alder Reactions of 5-R-1, 2, 4-Triazines under High Pressure Conditions

MI Savchuk, ES Starnovskaya, YK Shtaitz… - Russian Journal of …, 2018 - Springer
Synthesis of 5-Phenyl-2,2'-bipyridines 6-Substituted with Donor Groups by aza-Diels–Alder
Reactions of 5-R-1,2,4-Triazines u Page 1 2213 Synthesis of 5-Phenyl-2,2'-bipyridines 6-Substituted …

A facile synthesis of triazine integrated antipyrine derivatives through ecofriendly approach

A Rammohan, GM Reddy, AP Krinochkin… - Synthetic …, 2021 - Taylor & Francis
The present study describes a facile and solvent free synthesis of 1, 2, 4-triazine antipyrine
derivatives (2a–f) in prominent yields (70–85%) over nucleophilic substitution of 5 …

Recent advances in the synthesis of fluorinated compounds via an aryne intermediate

M Rahman, AK Bagdi, DS Kopchuk… - Organic & …, 2020 - pubs.rsc.org
The development of new methodologies for the synthesis of fluorinated organic molecules is
in high demand due to their wide applications in agriculture and pharmaceutical sciences …

One-step synthesis of 1, 4-bis (het) arylisoquinolines by the reaction of 1, 2, 4-triazines with arynes

DS Kopchuk, IL Nikonov, AF Khasanov… - Chemistry of …, 2019 - Springer
The reaction of 3, 6-bis (het) aryl-1, 2, 4-triazines (hetaryl≠ 2-pyridyl) with aryne
intermediates generated in situ was studied. As a result, novel 1, 4-bis (het) …