Flavone-C-glycosides from Cassia auriculata L. as possible inhibitors of phosphodiesterase-5 (PDE5): in vitro, molecular docking and molecular dynamics studies

A Ganapathy A, VM Hari Priya, K Baby… - Journal of …, 2024 - Taylor & Francis
Abstract Phosphodiesterase-5 (PDE5) is a homodimeric enzyme that specifically targets
cyclic guanosine monophosphate (cGMP), that mediates many downstream effects such as …

Effects of flavonoids on SARS–CoV–2 main protease (6W63): A molecular docking study

T Ertan-bolelli, K Bolelli… - Turkish …, 2023 - dergipark.org.tr
Public health is still under attack by a worldwide pandemic caused by a coronavirus which is
known to cause mainly respiratory and enteric disease in humans. Currently, still limited …

Computational approaches in the development of phosphodiesterase inhibitors

A Gaurav, M **ng, M Al‐Nema, A Gaurav… - Quantitative …, 2017 - books.google.com
Computational drug design tools have become indispensable in the quest for new drugs.
There is hardly any drug discovery program where computational methods are not …

Structural investigation of vesnarinone at the pore domains of open and open-inactivated states of hERG1 K+ channel

G Kayık, NŞ Tüzün, S Durdagi - Journal of Molecular Graphics and …, 2017 - Elsevier
In this study, the dynamics of vesnarinone bounded hERG1 K+ channels are investigated
using in silico approaches such as molecular docking, molecular dynamics (MD) …

[PDF][PDF] In silico design of hERG non-blocker compounds with retained pharmacological activity using multi-scale molecular modeling applications

G Kayık - 2017 - polen.itu.edu.tr
The subject of this Ph. D. thesis is to investigate the molecular interactions between hERG
blocker compounds and the central inner cavities of hERG K+ ion channels (in its open and …

[PDF][PDF] the body in movement: a clinical approach

M Probst, J Diedens - 2017 - lirias.kuleuven.be
Physiotherapy or body oriented therapy is often overlooked as an adjunctive treatment for
patients with eating disorders (ED). However, the integration of physiotherapy is based on …

[PDF][PDF] Aktuální možnosti a trendy v léčbě erektilní dysfunkce

MUDO Štanc - urologiepropraxi.cz
Erectile dysfunction (ED) is a very frequent disease. The past decades have witnessed a
dramatic development in its treatment, associated with an increased interest in this issue by …