Designing strategies, structural activity relationship and biological activity of recently developed nitrogen containing heterocyclic compounds as epidermal growth …

R Pal, G Teli, GSP Matada, PS Dhiwar - Journal of Molecular Structure, 2023‏ - Elsevier
Cancer cells have the ability of dysregulation and autonomous proliferation due to
unchecked production of definite molecules. These molecules are involved in the cell growth …

Poly (ADP-ribose) polymerase (PARP) inhibitors as anticancer agents: An outlook on clinical progress, synthetic strategies, biological activity, and structure-activity …

PK Das, GSP Matada, R Pal, L Maji, PS Dhiwar… - European journal of …, 2024‏ - Elsevier
Abstract Poly (ADP-ribose) polymerase (PARP) is considered an essential component in
case of DNA (Deoxyribonucleic acid) damage, response by sensing DNA damage and …

Therapeutic potential of anticancer activity of nitrogen-containing heterocyclic scaffolds as Janus kinase (JAK) inhibitor: Biological activity, selectivity, and structure …

R Pal, GSP Matada, G Teli, M Saha, R Patel - Bioorganic Chemistry, 2024‏ - Elsevier
The JAK-STAT signalling pathway is primarily involved in cytokine signalling and induces
various factors namely, erythropoietin, thrombopoietin, interferons, interleukins, and …

Nitrogen‐Containing Heterocyclic Scaffolds as EGFR Inhibitors: Design Approaches, Molecular Docking, and Structure‐Activity Relationships

R Pal, G Teli, G Swamy Purawarga Matada… - …, 2023‏ - Wiley Online Library
Cancer is a wide collection of diseases and among the numerous pathways involved in
cancer pathogenesis, pathway involving epidermal growth factor receptor (EGFR) is one of …

Benzothiazole a privileged scaffold for Cutting-Edges anticancer agents: Exploring drug design, structure-activity relationship, and docking studies

I Aayishamma, GSP Matada, R Pal, A Ghara… - European Journal of …, 2024‏ - Elsevier
Cancer is a major societal, public health, and economic burden in the 21 st century, with 9.7
million deaths in 2022 (9.96 million in 2020) and 20 million new cancer cases (19.6 million …

Design, synthesis, molecular docking and pharmacological evaluation of novel triazine-based triazole derivatives as potential anticonvulsant agents

AG Alhamzani, TA Yousef, MM Abou-Krisha… - Bioorganic & Medicinal …, 2022‏ - Elsevier
Triazine-linked triazole compounds (4a-j) were designed, synthesized, and then examined
for their anticonvulsant abilities. Compounds 4e, 4f, 4g, 4i, and 4j displayed significant …

Design, synthesis of 1, 2, 4-triazine derivatives as antidepressant and antioxidant agents: In vitro, in vivo and in silico studies

R Pal, B Kumar, GS PM, PA Chawla - Bioorganic Chemistry, 2023‏ - Elsevier
The novel series of substituted-N-(5, 6-diphenyl-1, 2, 4-triazin-3-yl) benzamides (R: 1–12)
were designed, synthesized and evaluated for in-vitro and in-vivo antidepressant-like …

Advancement of DDR1 and DDR2 Inhibitors: Therapeutic Potential of Bioactive Compounds, Designing Strategies, and Structure‐Activity Relationship (SAR)

R Pal, B Kumaraswamy, SK Md. Ashadul… - …, 2024‏ - Wiley Online Library
DDR1 and DDR2 are nonintegrin collagen receptors in the receptor tyrosine kinase family.
Both DDRs bind to various collagen types and perform crucial functions in embryo …

Synthesis of Novel Triazine-Based Chalcones and 8,9-dihydro-7H-pyrimido[4,5-b][1,4]diazepines as Potential Leads in the Search of Anticancer, Antibacterial and …

LM Moreno, J Quiroga, R Abonia, MP Crespo… - International Journal of …, 2024‏ - mdpi.com
This study presents the synthesis of four series of novel hybrid chalcones (20, 21) a–g and
(23, 24) a–g and six series of 1, 3, 5-triazine-based pyrimido [4, 5-b][1, 4] diazepines (28–33) …

Design, synthesis, and pharmacological evaluation of aryl oxadiazole linked 1, 2, 4-triazine derivatives as anticonvulsant agents

G Grover, R Pal, R Bhatia, MS Yar, R Nath… - Medicinal Chemistry …, 2022‏ - Springer
A series of new clubbed aryl oxadiazole-1, 2, 4-triazine derivatives (6a-l) were designed and
synthesized using appropriate chemical routes. The structures were designed to have the …