Cobalt and ruthenium complexes with pyrimidine based schiff base: Synthesis, characterization, anticancer activities and electrochemotherapy efficiency

ME Alkış, Ü Keleştemür, Y Alan, N Turan… - Journal of Molecular …, 2021 - Elsevier
In this study, a new Schiff base ligand and its two M (II) complexes [CoCl· L (H 2 O) 2]· 2H 2
O,[RuCl (p-cymene) L] were synthesized. The structural features were confirmed from their …

Halting colorectal cancer metastasis via novel dual nanomolar MMP-9/MAO-A quinoxaline-based inhibitors; design, synthesis, and evaluation

MS Ayoup, MM Abu-Serie, LF Awad, M Teleb… - European Journal of …, 2021 - Elsevier
Abstract Matrix metalloproteinase-9 (MMP-9) and monoamine oxidase-A (MAO-A) are
central signaling nodes in CRC and promotors of distant metastasis associated with high …

Synthesis, characterization, antiproliferative of pyrimidine based ligand and its Ni (II) and Pd (II) complexes and effectiveness of electroporation

ME Alkış, K Buldurun, N Turan, Y Alan… - Journal of …, 2022 - Taylor & Francis
In the study, a new Schiff base (ligand) was obtained using 4-aminopyrimidine-2 (1 H)-one,
the starting material, and 2, 3, 4-trimethoxy benzaldehyde. Ni (II) and Pd (II) complexes were …

Synthesis, spectroscopic characterization of novel phthalimides derivatives bearing a 1, 2, 3-triazole unit and examination as potential SARS-CoV-2 inhibitors via in …

A Tan - Journal of Molecular Structure, 2022 - Elsevier
In the present study, novel phthalimide derivatives 8 (af) and 9 (af) bearing a 1, 2, 3-triazole
subunit were synthesized via CuAAC reactions and characterized by 1 H, 13 C NMR, HR …

Novel hybrid isoindole‐1,3(2H)‐dione compounds containing a 1H‐tetrazole moiety: Synthesis, biological evaluation, and molecular docking studies

A Tan, S Kizilkaya, SAA Noma, B Ates… - Journal of biochemical …, 2022 - Wiley Online Library
In this study, novel hybrid isoindole‐1, 3 (2H)‐dione compounds (10 and 11) carrying a 1H‐
tetrazole moiety were synthesized, characterized and their inhibitory properties against …

Substituent effects in the formation of a few acenaphthenone-2-ylidene ketones and their molecular docking studies and in silico ADME profile

D Kuriakose, RK Thumpakara, A Jesna… - Journal of Molecular …, 2021 - Elsevier
We observed intriguing substituent effects in the reaction between 4-substituted
acetophenones and acenaphthenequinone in the presence of KOH in methanol. In all …

Design, Synthesis, and Docking Simulation of 1, 3, 4-Thiadiazolyl-Isoindole Thioglycosides and Hydrazinyl Sugar Analogs as Potential Anticancer Agents Targeting …

A El-Enazy, MN El-Bayaa, WI El-Sofany… - Polycyclic Aromatic …, 2024 - Taylor & Francis
The development of efficient strategies for overcoming cancer remains a standing objective
in medicinal chemistry. Design and synthesis of new potent compounds contribute efficiently …

Investigation of cytotoxic properties of some isoindole-related compounds bearing silyl and azide groups with in vitro and in silico studies

A Tan, A Köse, D Mete, G Şanlı-Mohamed… - … , Sulfur, and Silicon …, 2023 - Taylor & Francis
This study aims to evaluate the synthesis of isoindole-1, 3-dione analogues and their
cytotoxic potential. A549 and HeLa cells exposed to 250–100–50–25 µM doses of each …

Synthesis, Characterization, and Biological Evaluation of Some Isoindole‐1, 3‐(2H) Dione Derivatives

M Jabbour, MA Al-Khayat - Journal of Chemistry, 2023 - Wiley Online Library
In this study, we have established promising drug candidates with approved antimicrobial,
antioxidant, antileishmanial, and anticancer activities. We hereby report drug likeliness …

[PDF][PDF] MOLECULAR DOCKING STUDIES OF 3ꞌ, 5ꞌ-DICHOLORO-2ꞌ-HYDROXYACETOPHENONE-3-METHOXYBENZHYDRAZONE HYDRATE TOWARDS 1JXA …

D Kuriakose, MRP Kurup - Xaverian Research Journal - stxaviersaluva.ac.in
MOLECULAR DOCKING STUDIES OF 3ꞌ, 5ꞌ-DICHOLORO-2ꞌ-HYDROXYACETOPHENONE-3-METHOXYBENZHYDRAZONE
HYDRATE TOWARDS 1JXA RECEPTOR PROTEIN Page 58 DISCOURSE Xaverian …