Toward enzyme-responsive polymersome drug delivery

BC Paruchuri, V Gopal, S Sarupria, J Larsen - Nanomedicine, 2021 - Taylor & Francis
In drug delivery, enzyme-responsive drug carriers are becoming increasingly relevant
because of the growing association of disease pathology with enzyme overexpression …

Computational modeling of carbohydrate processing enzymes reactions

F Mendoza, L Masgrau - Current Opinion in Chemical Biology, 2021 - Elsevier
Carbohydrate processing enzymes are of biocatalytic interest. Glycoside hydrolases and the
recently discovered lytic polysaccharide monooxygenase for their use in biomass …

The hydrolysis mechanism of a GH45 cellulase and its potential relation to lytic transglycosylase and expansin function

VS Bharadwaj, BC Knott, J Ståhlberg… - Journal of Biological …, 2020 - ASBMB
Family 45 glycoside hydrolases (GH45) are endoglucanases that are integral to cellulolytic
secretomes, and their ability to break down cellulose has been successfully exploited in …

ATESA: an automated aimless shooting workflow

T Burgin, S Ellis, HB Mayes - Journal of Chemical Theory and …, 2022 - ACS Publications
Transition path sampling methods are powerful tools for studying the dynamics of rare
events in molecular simulations. However, these methods are generally restricted to experts …

Click-chemistry-based free Azide versus azido sugar detection enables rapid in vivo screening of Glycosynthase activity

A Agrawal, CK Bandi, T Burgin, Y Woo… - ACS chemical …, 2021 - ACS Publications
Engineering of carbohydrate-active enzymes such as glycosynthases to enable
chemoenzymatic synthesis of bespoke oligosaccharides has been limited by the lack of …

Mechanistic insight into the synthesis of fucooligosaccharides by α-L-fucosidase from Thermotoga maritima belonging to the GH29 family: in silico study

ME Pavón-Chimal, C Jiménez-Pérez… - Biologia, 2023 - Springer
In recent years, the synthesis of human milk oligosaccharides, particularly
fucooligosaccharides, has been investigated. These oligosaccharides provide protection …

Quick and Accurate Estimates of Mutation Effects on Transition-State Stabilization of Enzymes from Molecular Simulations with Restrained Transition States

T Burgin, J Pfaendtner, DAC Beck - The Journal of Physical …, 2022 - ACS Publications
Data science and machine learning are revolutionizing enzyme engineering; however, high-
throughput simulations for screening large libraries of enzyme variants remain a challenge …

High-throughput screening of glycosynthases using azido sugars for oligosaccharides synthesis

M Kumar, CK Bandi, SPS Chundawat - Methods in Enzymology, 2023 - Elsevier
Glycosynthases are mutant glycosyl hydrolases that can synthesize glycosidic bonds
between acceptor glycone/aglycone groups and activated donor sugars with suitable …

Click-chemistry enabled directed evolution of glycosynthases for bespoke glycans synthesis

A Agrawal, CK Bandi, T Burgin, Y Woo, HB Mayes… - bioRxiv, 2020 - biorxiv.org
Engineering of carbohydrate-active enzymes like glycosynthases for chemoenzymatic
synthesis of bespoke oligosaccharides has been limited by the lack of suitable directed …

Machine learning assisted ligand binding energy prediction for in silico generated glycosyl hydrolase enzyme combinatorial mutant library

I Guranovic, M Kumar, CK Bandi, SPS Chundawat - bioRxiv, 2022 - biorxiv.org
Molecular docking is a computational method used to predict the preferred binding
orientation of one molecule to another when bound to each other to form an energetically …